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7-TM Receptors
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ICI 185,282
ICI 185,282 is a potent thromboxane receptor antagonist. Learn MoreStarting at: $95.00
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L-798,106
L-798,106 is a potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2 respectively). Learn MoreStarting at: $140.00
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TCS 2510
TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM), which displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM. Learn MoreStarting at: $139.00
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AA 2414
AA 2414 is a thromboxane A2 (TP) receptor antagonist, which inhibits platelet aggregation and bronchoconstriction induced by a TXA2 mimetic in guinea pigs. Learn MoreStarting at: $90.00
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Iloprost
Iloprost is a prostacyclin (PGI2) analog that inhibits platelet aggregation induced by collagen, thrombin and ADP with IC50 values of 0.24, 0.71 and 1.07 nM respectively. Learn MoreStarting at: $239.00
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Ozagrel hydrochloride
Ozagrel hydrochloride is a potent and selective inhibitor of thromboxane (TXA2) synthetase that inhibits platelet aggregation in vitro and arachidonate-induced arterial contraction in vivo. Learn MoreStarting at: $85.00
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Epoprostenol
Epoprostenol is a endogenous prostanoid that is a potent agonist at IP prostanoid receptors. Learn MoreStarting at: $389.00
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Sulprostone
Sulprostone is a selective EP3 and EP1 receptor agonist and also is synthetic PGE2 analog and allodynic agent. Learn MoreStarting at: $119.00
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Misoprostol
Misoprostol is a cytoprotective prostaglandin E1 analog with Ki values of 120, 250, 67 and 67 nM at cloned mouse EP1, EP2, EP3 and EP4 receptors respectively. Learn MoreStarting at: $99.00
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U 46619
U 46619 is a stable synthetic analog of the endoperoxide prostaglandin PGH2 first prepared in 1975, and acts as a thromboxane A2 (TP) receptor agonist. Learn MoreStarting at: $109.00
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(+)-Fluprostenol
(+)-Fluprostenol, a prostaglandin F2α (FP) receptor agonist, stimulates intracellular calcium mobilization in cloned human ocular FP receptors, rat A7r5 cells and mouse 3T3 cells (EC50 values are 17.5, 19.1 and 37.3 nM respectively). Learn MoreStarting at: $55.00
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GW 627368
GW 627368 is a selective prostanoid EP4 receptor competitive antagonist with additional affinity at TP receptors (pKi values are 7.0 and 6.8 in competition radioligand bioassays). Learn MoreStarting at: $179.00
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16,16-Dimethyl Prostaglandin E2
16,16-Dimethyl Prostaglandin E2 is a synthetic derivative of prostaglandin E2, which increases embryonic stem cell (ESC) hematopoietic colony formation in mouse bone marrow. Learn MoreStarting at: $85.00
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Prostaglandin F2α
Prostaglandin E2 and F2α receptor agonist. Naturally-occurring prostaglandin and potent vasoconstrictor. Learn MoreStarting at: $159.00
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WAY 267464 dihydrochloride
WAY 267464 dihydrochloride is a potent, selective non-peptide oxytocin receptor (OTR) agonist. Learn MoreStarting at: $189.00
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L-371,257
RWJ 50271 is a selective inhibitor of LFA-1 (lymphocyte function-associated antigen-1) adhesion to soluble intercellular adhesion molecule (sICAM) (IC50 = 5 μM in HL60 cells). Learn MoreStarting at: $155.00
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L-368,899 hydrochloride
L-368,899 hydrochloride is a potent, non-peptide and orally active oxytocin receptor antagonist (IC50 = 8.9 nM) that displays > 40-fold selectivity over vasopressin V1a and V2 receptors (IC50 values are 370 and 570 nM respectively). Learn MoreStarting at: $90.00
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WEB 2086
WEB 2086 is a potent, selective platelet-activating factor (PAF) receptor antagonist (Ki = 16.3 nM). Which inhibits growth and proliferation of MCF-7 breast cancer cells. Learn MoreStarting at: $75.00
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PCA 4248
PCA 4248 is a specific PAF antagonist,which inhibits rabbit platelet aggregation with an IC50 value of 1.05 μM and has no significant activity on Ca2+ channels. Learn MoreStarting at: $90.00
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PAF (C16)
PAF (C16) is an endogenous platelet-activating factor (PAF) and ligand for PAF receptors. Learn MoreStarting at: $150.00
