Histamine H2 Receptors
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Zolantidine dimaleate
Zolantidine dimaleate is a potent, selective and brain penetrating H2 receptor antagonist. Learn MoreStarting at: $100.00
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Aminopotentidine
Aminopotentidine is a H2 antagonist (KB values are 220 and 280 nM at human and guinea pig H2 receptors respectively) and precursor for the synthesis of the [125I]-iodo derivative. Learn MoreStarting at: $115.00
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Amthamine dihydrobromide
Amthamine dihydrobromide is a highly selective H2 agonist, slightly more potent than histamine itself. It induces vasodilation of cerebral arteries and decreases myogenic tone in vitro. Learn MoreStarting at: $95.00
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Dimaprit dihydrochloride
Dimaprit dihydrochloride is a selective H2 agonist with central effects upon systemic administration, which also inhibits nNOS (IC50 = 49 μM). Learn MoreStarting at: $90.00
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Burimamide oxalate
Burimamide oxalate is a histamine H3/H2 receptor antagonist (Ki values are 0.07, 7.8 and 290 μM for H3, H2 and H1 receptors respectively), which displays partial agonist activity in SK-N-MC cells and produces antinociceptive effects following intraventricular administration (ED50 = 183 nmol/mouse in hot-plate test). Learn MoreStarting at: $115.00
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Ranitidine hydrochloride
Ranitidine hydrochloride is a potent, selective and competitive histamine H2 receptor antagonist that inhibits gastric acid secretion induced by histamine, pentagastrin, bethanecol and food in vivo. Learn MoreStarting at: $39.00
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Tiotidine
Tiotidine is a potent histamine H2-receptor antagonist with negligible activity against H1- and H3- receptors. Learn MoreStarting at: $59.00
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ICI 162846
ICI 162846 is a potent histamine H2 receptor antagonist. Learn MoreStarting at: $109.00