Estrogen (GPR30) Receptors

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  • G-15

    G-15 is a high affinity and selective GPR30 receptor antagonist (Ki = 20 nM) that displays no affinity for ERα and ERβ at concentrations up to 10 μM. Learn More

    Starting at: $120.00

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  • G-36

    G-36 is an antagonist of GPR30 which selectively inhibits estrogen-mediated activation of PI3-K by GPR30. Learn More

    Starting at: $135.00

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  • G-1

    G-1 is a potent and selective GPR30 receptor agonist that increases cytosolic Ca2+ and inhibits migration of SKBr3 cells and MCF-7 cells in response to chemoattractants with IC50 values of 0.7 and 1.6 nM respectively in vitro. Learn More

    Starting at: $139.00

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3 Item(s)

per page