Esterases

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  • HA 130

    HA 130 is a selective autotaxin inhibitor (IC50 = 28 nM), which binds and inhibits autotaxin reversibly. Learn More

    Starting at: $135.00

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  • S 32826

    S 32826 is an inhibitor of autotaxin (IC50 = 9 nM), which displays similar inhibitory effects at all three autotaxin isoforms (α, β and γ)and inhibits LPA release from adipocytes (IC50 = 90 nM). Learn More

    Starting at: $135.00

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  • Pristimerin

    Pristimerin is a potent and reversible inhibitor of monoacylglycerol lipase (MGL) (IC50 = 93 nM), which displays antitumor, anti-inflammatory and antimicrobial activities. Learn More

    Starting at: $135.00

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  • GSK 264220A

    GSK 264220A is an endothelial lipase and lipoprotein lipase inhibitor with IC50 values of 0.13 and 0.10 μM respectively. Learn More

    Starting at: $119.00

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  • RHC 80267

    RHC 80267 is an inhibitor of diacylglycerol lipase that potentiates acetylcholine evoked relaxation in mesenteric arteries by the inhibition of cholinesterase activity. Learn More

    Starting at: $99.00

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  • Tacrine hydrochloride

    AIDA is a relatively potent and selective antagonist of group I metabotropic glutamate receptors (mGlu1a), having no effect on group II (mGlu2) or group III (mGlu4) receptors expressed individually in baby hamster kidney cells. Learn More

    Starting at: $60.00

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  • Ambenonium dichloride

    Ambenonium dichloride is a extremely potent, selective and rapidly reversible inhibitor of acetylcholinesterase (AChE) with IC50 values =0.000698 and 8.20 μM at AChE and BChE respectively. Learn More

    Starting at: $99.00

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  • Acephate

    Anticholinesterase insecticide that produces cholinotoxicity, which displays weak inhibition of rat acetylcholinesterase (AChE) but potently inhibits cockroach AChE. Learn More

    Starting at: $59.00

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  • Physostigmine hemisulfate

    Physostigmine hemisulfate is a cholinesterase inhibitor. Learn More

    Starting at: $33.00

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  • Galanthamine hydrobromide

    Galanthamine hydrobromide is a long-acting, centrally active acetylcholinesterase inhibitor (IC50 = 410 nM) and allosteric potentiator at neuronal nicotinic ACh receptors. Learn More

    Starting at: $75.00

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  • Rivastigmine tartrate

    Rivastigmine tartrate is a dual cholinesterase inhibitor (ChEI) which inhibits both butyrylcholinesterase (BChE) and acetylcholinesterase (AChE). Learn More

    Starting at: $70.00

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  • PE 154

    PE 154 is a potent fluorescent inhibitor of human acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) (IC50 values are 280 pM and 16 nM respectively), which targets and labels β-amyloid plaques in histochemical analysis. Learn More

    Starting at: $160.00

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  • Phenserine

    Phenserine is a Physostigmine analog that inhibits acetylcholinesterase.Phenserin also inhibits production of amyloid precursor protein (APP) and A&beta and improves morris water maze performance of scopolamine-treated rats. Learn More

    Starting at: $95.00

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  • STF 083010

    STF 083010 is an inhibitor of IRE1α endonuclease activity; blocks endogenous XBP1 mRNA splicing. Learn More

    Starting at: $119.00

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  • Edelfosine

    Edelfosine is a synthetic lysophospholipid analog that selectively inhibits phosphatidylinositol phospholipase C. Learn More

    Starting at: $89.00

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  • LY 311727

    AM 630 is a CB2 antagonist/inverse agonist (Ki = 31.2 nM) that displays 165-fold selectivity over CB1 receptors. Learn More

    Starting at: $140.00

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  • o-3M3FBS

    o-3M3FBS is an inactive analog of m-3M3FBS. Used as a negative control. Learn More

    Starting at: $99.00

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  • OBAA

    OBAA is a potent inhibitor of phospholipase A2 (IC50 = 70 nM), which reduces bronchospasm in guinea pigs in vivo. Learn More

    Starting at: $90.00

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  • m-3M3FBS

    m-3M3FBS is a activator of phospholipase C (PLC), which stimulates superoxide generation, Ca2+ release and inositol phosphate formation in a variety of cell types, and inhibits growth of the leukemic cell lines U937 and THP-1. Learn More

    Starting at: $98.00

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  • AACOCF3

    AACOCF3 is an inhibitor of cytosolic (85 kDa) phospholipase A2. It also inhibits fatty acid amide hydrolase (FAAH, anandamide amidase) in vitro. Learn More

    Starting at: $65.00

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