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Esterases
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S 32826
S 32826 is an inhibitor of autotaxin (IC50 = 9 nM), which displays similar inhibitory effects at all three autotaxin isoforms (α, β and γ)and inhibits LPA release from adipocytes (IC50 = 90 nM). Learn MoreStarting at: $135.00
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HA 130
HA 130 is a selective autotaxin inhibitor (IC50 = 28 nM), which binds and inhibits autotaxin reversibly. Learn MoreStarting at: $135.00
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Pristimerin
Pristimerin is a potent and reversible inhibitor of monoacylglycerol lipase (MGL) (IC50 = 93 nM), which displays antitumor, anti-inflammatory and antimicrobial activities. Learn MoreStarting at: $135.00
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GSK 264220A
GSK 264220A is an endothelial lipase and lipoprotein lipase inhibitor with IC50 values of 0.13 and 0.10 μM respectively. Learn MoreStarting at: $119.00
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RHC 80267
RHC 80267 is an inhibitor of diacylglycerol lipase that potentiates acetylcholine evoked relaxation in mesenteric arteries by the inhibition of cholinesterase activity. Learn MoreStarting at: $99.00
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Ambenonium dichloride
Ambenonium dichloride is a extremely potent, selective and rapidly reversible inhibitor of acetylcholinesterase (AChE) with IC50 values =0.000698 and 8.20 μM at AChE and BChE respectively. Learn MoreStarting at: $99.00
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Tacrine hydrochloride
AIDA is a relatively potent and selective antagonist of group I metabotropic glutamate receptors (mGlu1a), having no effect on group II (mGlu2) or group III (mGlu4) receptors expressed individually in baby hamster kidney cells. Learn MoreStarting at: $60.00
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Acephate
Anticholinesterase insecticide that produces cholinotoxicity, which displays weak inhibition of rat acetylcholinesterase (AChE) but potently inhibits cockroach AChE. Learn MoreStarting at: $59.00
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Rivastigmine tartrate
Rivastigmine tartrate is a dual cholinesterase inhibitor (ChEI) which inhibits both butyrylcholinesterase (BChE) and acetylcholinesterase (AChE). Learn MoreStarting at: $70.00
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PE 154
PE 154 is a potent fluorescent inhibitor of human acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) (IC50 values are 280 pM and 16 nM respectively), which targets and labels β-amyloid plaques in histochemical analysis. Learn MoreStarting at: $160.00
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Phenserine
Phenserine is a Physostigmine analog that inhibits acetylcholinesterase.Phenserin also inhibits production of amyloid precursor protein (APP) and A&beta and improves morris water maze performance of scopolamine-treated rats. Learn MoreStarting at: $95.00
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Galanthamine hydrobromide
Galanthamine hydrobromide is a long-acting, centrally active acetylcholinesterase inhibitor (IC50 = 410 nM) and allosteric potentiator at neuronal nicotinic ACh receptors. Learn MoreStarting at: $75.00
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Physostigmine hemisulfate
Physostigmine hemisulfate is a cholinesterase inhibitor. Learn MoreStarting at: $33.00
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STF 083010
STF 083010 is an inhibitor of IRE1α endonuclease activity; blocks endogenous XBP1 mRNA splicing. Learn MoreStarting at: $119.00
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VU 0155069
VU 0155069 is a potent and selective phospholipase D1 (PLD1) inhibitor (IC50 values are 46 and 933 nM for PLD1 and PLD2 respectively), which inhibits migration of human and mouse breast cancer cell lines in transwell assays. Learn MoreStarting at: $130.00
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Edelfosine
Edelfosine is a synthetic lysophospholipid analog that selectively inhibits phosphatidylinositol phospholipase C. Learn MoreStarting at: $89.00
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LY 311727
AM 630 is a CB2 antagonist/inverse agonist (Ki = 31.2 nM) that displays 165-fold selectivity over CB1 receptors. Learn MoreStarting at: $140.00
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o-3M3FBS
o-3M3FBS is an inactive analog of m-3M3FBS. Used as a negative control. Learn MoreStarting at: $99.00
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OBAA
OBAA is a potent inhibitor of phospholipase A2 (IC50 = 70 nM), which reduces bronchospasm in guinea pigs in vivo. Learn MoreStarting at: $90.00
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m-3M3FBS
m-3M3FBS is a activator of phospholipase C (PLC), which stimulates superoxide generation, Ca2+ release and inositol phosphate formation in a variety of cell types, and inhibits growth of the leukemic cell lines U937 and THP-1. Learn MoreStarting at: $98.00
