Esterases
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AACOCF3
AACOCF3 is an inhibitor of cytosolic (85 kDa) phospholipase A2. It also inhibits fatty acid amide hydrolase (FAAH, anandamide amidase) in vitro. Learn MoreStarting at: $65.00
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YM 26734
YM 26734 is a competitive inhibitor of secretory phospholipase A2 (sPLA2) that exhibits a broad inhibitory profile to several sPLA2s (IC50 values are 0.2, 1, 1, 1 and 3 μM for sPLA2-X, -IIA, -IID, -V and -IIE respectively). Learn MoreStarting at: $135.00
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U 73343
U 73343 is an inactive analog of U 73122. Can be used as a negative control. Learn MoreStarting at: $85.00
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PACOCF3
PACOCF3 is a phospholipase A2 inhibitor. Can also alter Ca2+ signaling in renal tubular cells. Learn MoreStarting at: $75.00
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VU 0364739 hydrochloride
VU 0364739 hydrochloride is a potent and selective phospholipase D2 (PLD2) inhibitor (IC50 = 20 nM) which displays 75-fold selectivity against PLD1 (IC50 = 1500 nM). Learn MoreStarting at: $155.00
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SGC-CBP30
SGC-CBP30 is a potent CREBBP/EP300 bromodomain inhibitor (IC50 values are 21-69 and 38 nM for CREBBP and EP300 bromodomains respectively), which displays over 40-fold selectivity for CREBBP over BRD4(1). Learn MoreStarting at: $199.00