Adenosine Receptors

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  • 2-Chloro-N6-cyclopentyladenosine

    2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 0.8, 2300 and 42 nM for human A1, A2A and A3 receptors respectively; EC50 = 18800 nM for hA2B). Learn More

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  • N6-Cyclopentyladenosine

    N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 2.3, 790 and 43 nM for human A1, A2A and A3 receptors respectively; EC50 = 18600 nM for hA2B). Learn More

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  • PSB 36

    PSB 36 is a Potent and selective A1 adenosine receptor antagonist with binding affinities of 0.12, 187, 552, 6500 and 2300 nM for rA1, hA2B, rA2A, rA3 and hA3 receptors respectively. Learn More

    Starting at: $129.00

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  • SLV 320

    SLV 320 is a potent and selective adenosine A1 receptor antagonist (Ki values are 1, 200, 398 and 3981 nM at human A1, A3, A2A and A2B receptors respectively). Learn More

    Starting at: $105.00

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  • 2'-MeCCPA

    2'-MeCCPA is a potent and highly selective agonist at A1 adenosine receptors (Ki values are 3.3, 9580, 37600 and 1150 nM for human recombinant A1, A2A, A2B and A3 receptors respectively), which acts as a full agonist and inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC50 value of 13.1 nM. Learn More

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  • 1,3-Dipropyl-8-phenylxanthine

    1,3-Dipropyl-8-phenylxanthine is a selective A1 adenosine antagonist. Learn More

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  • KW 3902

    KW 3902 is a selective adenosine A1 receptor antagonist; displays 890-fold selectivity for rat A1 receptors over A2A receptors (Ki values are 0.19 and 170 nM respectively). Learn More

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  • PD 81723

    PD 81723 is an allosteric potentiator at the adenosine A1 receptor which acts via agonist-dependent and -independent mechanisms. Learn More

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  • SDZ WAG 994

    SDZ WAG 994 is a potent and selective A1 adenosine receptor agonist (Ki values are 23, > 10000 and 25000 nM for A1, A2A and A2B receptors respectively). Learn More

    Starting at: $145.00

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  • DPCPX

    DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Learn More

    Starting at: $119.00

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  • (±)-5'-Chloro-5'-deoxy-ENBA

    (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist (Ki values are 0.51, 1290, 1340 and 2740 nM at A1, A3, A2A and A2B receptors respectively). Learn More

    Starting at: $135.00

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  • GR 79236

    GR 79236 is a adenosine A1 receptor agonist (Ki = 3.1 nM). Learn More

    Starting at: $155.00

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  • MRS 1754

    MRS 1754 is a selective adenosine A2B receptor antagonist (Ki values are 1.97, 16.8, 403, 503, 570 and 612 nM for hA2B, rA1, hA1, hA2A, hA3 and rA2A receptors respectively). Learn More

    Starting at: $139.00

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  • CV 1808

    CV 1808, a adenosine A2 receptor agonist, is coronary vasodilator, antihypertensive and antipsychotic following systemic administration in vivo. Learn More

    Starting at: $65.00

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  • PSB 603

    PSB 603 is an adenosine A2B receptor antagonist that displays > 17000-fold selectivity over other adenosine receptors (Ki values are 0.553, > 10000, > 10000 and > 10000 nM for A2B, A1, A2A and A3 receptors respectively). Learn More

    Starting at: $169.00

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  • BAY 60-6583

    BAY 60-6583 is a potent adenosine A2B receptor agonist that decreases fMLP-induced superoxide production in neutrophils at low concentrations (1-10 nM). Learn More

    Starting at: $139.00

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  • PSB 0788

    PSB 0788 is a potent and selective adenosine A2B receptor antagonist (IC50 = 3.64 nM at human A2B receptors) that displays > 100-fold selectivity over hA1, hA2A and hA3 receptors. Learn More

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  • PSB 1115

    PSB 1115 is a highly selective, water-soluble, human A2B adenosine receptor antagonist. Ki values are 53.4, > 10000 and > 10000 nM at human A2B, A1 and A3 receptors respectively. Learn More

    Starting at: $105.00

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  • MRS 1706

    MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist (Ki values are 1.39, 157, 112 and 230 nM for human A2B, A1, A2A and A3 receptors respectively). Learn More

    Starting at: $119.00

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  • SCH 58261

    2-Iminopiperidine hydrochloride is an inhibitor of NO synthases, more potent than NG-methyl-L-arginine and selective for iNOS. Learn More

    Starting at: $135.00

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