Adenosine Receptors
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DPCPX
DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Learn MoreStarting at: $119.00
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1,3-Dipropyl-8-phenylxanthine
1,3-Dipropyl-8-phenylxanthine is a selective A1 adenosine antagonist. Learn MoreStarting at: $95.00
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PSB 36
PSB 36 is a Potent and selective A1 adenosine receptor antagonist with binding affinities of 0.12, 187, 552, 6500 and 2300 nM for rA1, hA2B, rA2A, rA3 and hA3 receptors respectively. Learn MoreStarting at: $129.00
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N6-Cyclopentyladenosine
N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 2.3, 790 and 43 nM for human A1, A2A and A3 receptors respectively; EC50 = 18600 nM for hA2B). Learn MoreStarting at: $89.00
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2-Chloro-N6-cyclopentyladenosine
2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 0.8, 2300 and 42 nM for human A1, A2A and A3 receptors respectively; EC50 = 18800 nM for hA2B). Learn MoreStarting at: $99.00
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SLV 320
SLV 320 is a potent and selective adenosine A1 receptor antagonist (Ki values are 1, 200, 398 and 3981 nM at human A1, A3, A2A and A2B receptors respectively). Learn MoreStarting at: $105.00
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2'-MeCCPA
2'-MeCCPA is a potent and highly selective agonist at A1 adenosine receptors (Ki values are 3.3, 9580, 37600 and 1150 nM for human recombinant A1, A2A, A2B and A3 receptors respectively), which acts as a full agonist and inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC50 value of 13.1 nM. Learn MoreStarting at: $189.00
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KW 3902
KW 3902 is a selective adenosine A1 receptor antagonist; displays 890-fold selectivity for rat A1 receptors over A2A receptors (Ki values are 0.19 and 170 nM respectively). Learn MoreStarting at: $115.00
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PD 81723
PD 81723 is an allosteric potentiator at the adenosine A1 receptor which acts via agonist-dependent and -independent mechanisms. Learn MoreStarting at: $95.00
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SDZ WAG 994
SDZ WAG 994 is a potent and selective A1 adenosine receptor agonist (Ki values are 23, > 10000 and 25000 nM for A1, A2A and A2B receptors respectively). Learn MoreStarting at: $145.00
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GR 79236
GR 79236 is a adenosine A1 receptor agonist (Ki = 3.1 nM). Learn MoreStarting at: $155.00
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(±)-5'-Chloro-5'-deoxy-ENBA
(±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist (Ki values are 0.51, 1290, 1340 and 2740 nM at A1, A3, A2A and A2B receptors respectively). Learn MoreStarting at: $135.00
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BAY 60-6583
BAY 60-6583 is a potent adenosine A2B receptor agonist that decreases fMLP-induced superoxide production in neutrophils at low concentrations (1-10 nM). Learn MoreStarting at: $139.00
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CV 1808
CV 1808, a adenosine A2 receptor agonist, is coronary vasodilator, antihypertensive and antipsychotic following systemic administration in vivo. Learn MoreStarting at: $65.00
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PSB 1115
PSB 1115 is a highly selective, water-soluble, human A2B adenosine receptor antagonist. Ki values are 53.4, > 10000 and > 10000 nM at human A2B, A1 and A3 receptors respectively. Learn MoreStarting at: $105.00
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MRS 1754
MRS 1754 is a selective adenosine A2B receptor antagonist (Ki values are 1.97, 16.8, 403, 503, 570 and 612 nM for hA2B, rA1, hA1, hA2A, hA3 and rA2A receptors respectively). Learn MoreStarting at: $139.00
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MRS 1706
MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist (Ki values are 1.39, 157, 112 and 230 nM for human A2B, A1, A2A and A3 receptors respectively). Learn MoreStarting at: $119.00
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PSB 603
PSB 603 is an adenosine A2B receptor antagonist that displays > 17000-fold selectivity over other adenosine receptors (Ki values are 0.553, > 10000, > 10000 and > 10000 nM for A2B, A1, A2A and A3 receptors respectively). Learn MoreStarting at: $169.00
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PSB 0788
PSB 0788 is a potent and selective adenosine A2B receptor antagonist (IC50 = 3.64 nM at human A2B receptors) that displays > 100-fold selectivity over hA1, hA2A and hA3 receptors. Learn MoreStarting at: $115.00
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NPEC-caged-D-AP5
NPEC-caged-D-AP5 is a D-AP5 caged with the photosensitive 1-(2-nitrophenyl)ethoxycarbonyl (NPEC) group. NMDA receptor antagonist. Learn MoreStarting at: $189.00