Adenosine A3 Receptors

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  • MRS 3777 hemioxalate

    MRS 3777 hemioxalate is a high affinity adenosine A3 receptor antagonist (Ki = 47 nM) that displays > 200-fold selectivity versus A1, A2A and A2B receptors. Learn More

    Starting at: $100.00

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  • MRS 1220

    MRS 1220 is a potent and highly selective antagonist at the human A3 adenosine receptor (Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. Learn More

    Starting at: $135.00

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  • MRS 1334

    MRS 1334 is a potent and highly selective antagonist for the human adenosine A3 receptor. Ki values are 2.69 nM at hA3, and > 100 μM at rat A1 and rat A2A receptors. Learn More

    Starting at: $110.00

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  • MRE 3008F20

    MRE 3008F20 is a potent adenosine A3 receptor competitive antagonist, which potently inhibits agonist-induced cyclic AMP elevation in resting T lymphocytes (IC50 = 5 nM). Learn More

    Starting at: $135.00

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  • VUF 5574

    VUF 5574 is a potent, selective, competitive antagonist for the human adenosine A3 receptor (Ki = 4 nM), which displays ≥ 2500-fold selectivity over A1 and A2A receptors. Learn More

    Starting at: $109.00

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  • HEMADO

    HEMADO is an high affinity and selective adenosine A3 receptor agonist (Ki values are 1.1, 327, 1230 and > 30,000 nM for human A3, A1, A2A and A2B receptors respectively). Learn More

    Starting at: $139.00

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  • PSB 11 hydrochloride

    PSB 11 hydrochloride is a potent and selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor (Ki values are 2.3 and > 10000 nM respectively), which displays > 1000-fold selectivity over human A1 and A2A receptors (Ki values are 4.1 and 3.3 μM respectively) and > 180-fold selectivity over rat A1, rat A2A and mouse A2B receptors. Learn More

    Starting at: $139.00

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  • PSB 10 hydrochloride

    PSB 10 hydrochloride is potent and highly selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor. Learn More

    Starting at: $129.00

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