Adenosine Receptors
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ANR 94
ANR 94 is an Adenosine A2A receptor (AA2AR) antagonist with Ki values of 643 and 46 nM for rat and human AA2ARs respectively. Learn MoreStarting at: $139.00
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SCH 58261
2-Iminopiperidine hydrochloride is an inhibitor of NO synthases, more potent than NG-methyl-L-arginine and selective for iNOS. Learn MoreStarting at: $135.00
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PSB 10 hydrochloride
PSB 10 hydrochloride is potent and highly selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor. Learn MoreStarting at: $129.00
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PSB 11 hydrochloride
PSB 11 hydrochloride is a potent and selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor (Ki values are 2.3 and > 10000 nM respectively), which displays > 1000-fold selectivity over human A1 and A2A receptors (Ki values are 4.1 and 3.3 μM respectively) and > 180-fold selectivity over rat A1, rat A2A and mouse A2B receptors. Learn MoreStarting at: $139.00
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HEMADO
HEMADO is an high affinity and selective adenosine A3 receptor agonist (Ki values are 1.1, 327, 1230 and > 30,000 nM for human A3, A1, A2A and A2B receptors respectively). Learn MoreStarting at: $139.00
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VUF 5574
VUF 5574 is a potent, selective, competitive antagonist for the human adenosine A3 receptor (Ki = 4 nM), which displays ≥ 2500-fold selectivity over A1 and A2A receptors. Learn MoreStarting at: $109.00
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MRE 3008F20
MRE 3008F20 is a potent adenosine A3 receptor competitive antagonist, which potently inhibits agonist-induced cyclic AMP elevation in resting T lymphocytes (IC50 = 5 nM). Learn MoreStarting at: $135.00
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MRS 1334
MRS 1334 is a potent and highly selective antagonist for the human adenosine A3 receptor. Ki values are 2.69 nM at hA3, and > 100 μM at rat A1 and rat A2A receptors. Learn MoreStarting at: $110.00
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MRS 1220
MRS 1220 is a potent and highly selective antagonist at the human A3 adenosine receptor (Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. Learn MoreStarting at: $135.00
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MRS 3777 hemioxalate
MRS 3777 hemioxalate is a high affinity adenosine A3 receptor antagonist (Ki = 47 nM) that displays > 200-fold selectivity versus A1, A2A and A2B receptors. Learn MoreStarting at: $100.00
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XCC
XCC is an adenosine receptor antagonist (Ki values are 42, 68 and 1130 nM for A1, A2B and A2A receptors). Learn MoreStarting at: $95.00
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NECA
NECA is a potent adenosine receptor agonist (Ki values are 14, 20 and 6.2 nM for human A1, A2A and A3 receptors respectively; EC50 = 2.4 μM for human A2B), which inhibits platelet aggregation and is centrally active in vivo. Learn MoreStarting at: $49.00
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CGH 2466 dihydrochloride
Adenosine A1, A2B and A3 receptor antagonist (IC50 values are 19, 21, and 80 nM respectively). Also inhibits p38 MAPK (IC50 = 187 - 400 nM) and phosphodiesterase type 4D (IC50 = 22 nM). Learn MoreStarting at: $99.00
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2-Chloroadenosine
2-Chloroadenosine is a metabolically stable analog of adenosine that behaves as an adenosine receptor agonist (Ki values are 300, 80 and 1900 nM for A1, A2A and A3 receptors respectively). Learn MoreStarting at: $75.00
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Caffeine
Caffeine is a central nervous system stimulant, which mobilizes calcium from intracellular stores and inhibits benzodiazepine binding to GABA receptors. Learn MoreStarting at: $69.00
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XAC
XAC is an adenosine receptor antagonist (IC50 values are 1.8 and 114 nM at A1 and A2 receptors respectively). Learn MoreStarting at: $95.00