Adenosine Receptors

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  • ANR 94

    ANR 94 is an Adenosine A2A receptor (AA2AR) antagonist with Ki values of 643 and 46 nM for rat and human AA2ARs respectively. Learn More

    Starting at: $139.00

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  • SCH 58261

    2-Iminopiperidine hydrochloride is an inhibitor of NO synthases, more potent than NG-methyl-L-arginine and selective for iNOS. Learn More

    Starting at: $135.00

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  • PSB 10 hydrochloride

    PSB 10 hydrochloride is potent and highly selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor. Learn More

    Starting at: $129.00

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  • PSB 11 hydrochloride

    PSB 11 hydrochloride is a potent and selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor (Ki values are 2.3 and > 10000 nM respectively), which displays > 1000-fold selectivity over human A1 and A2A receptors (Ki values are 4.1 and 3.3 μM respectively) and > 180-fold selectivity over rat A1, rat A2A and mouse A2B receptors. Learn More

    Starting at: $139.00

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  • HEMADO

    HEMADO is an high affinity and selective adenosine A3 receptor agonist (Ki values are 1.1, 327, 1230 and > 30,000 nM for human A3, A1, A2A and A2B receptors respectively). Learn More

    Starting at: $139.00

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  • VUF 5574

    VUF 5574 is a potent, selective, competitive antagonist for the human adenosine A3 receptor (Ki = 4 nM), which displays ≥ 2500-fold selectivity over A1 and A2A receptors. Learn More

    Starting at: $109.00

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  • MRE 3008F20

    MRE 3008F20 is a potent adenosine A3 receptor competitive antagonist, which potently inhibits agonist-induced cyclic AMP elevation in resting T lymphocytes (IC50 = 5 nM). Learn More

    Starting at: $135.00

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  • MRS 1334

    MRS 1334 is a potent and highly selective antagonist for the human adenosine A3 receptor. Ki values are 2.69 nM at hA3, and > 100 μM at rat A1 and rat A2A receptors. Learn More

    Starting at: $110.00

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  • MRS 1220

    MRS 1220 is a potent and highly selective antagonist at the human A3 adenosine receptor (Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. Learn More

    Starting at: $135.00

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  • MRS 3777 hemioxalate

    MRS 3777 hemioxalate is a high affinity adenosine A3 receptor antagonist (Ki = 47 nM) that displays > 200-fold selectivity versus A1, A2A and A2B receptors. Learn More

    Starting at: $100.00

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  • XCC

    XCC is an adenosine receptor antagonist (Ki values are 42, 68 and 1130 nM for A1, A2B and A2A receptors). Learn More

    Starting at: $95.00

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  • NECA

    NECA is a potent adenosine receptor agonist (Ki values are 14, 20 and 6.2 nM for human A1, A2A and A3 receptors respectively; EC50 = 2.4 μM for human A2B), which inhibits platelet aggregation and is centrally active in vivo. Learn More

    Starting at: $49.00

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  • CGH 2466 dihydrochloride

    Adenosine A1, A2B and A3 receptor antagonist (IC50 values are 19, 21, and 80 nM respectively). Also inhibits p38 MAPK (IC50 = 187 - 400 nM) and phosphodiesterase type 4D (IC50 = 22 nM). Learn More

    Starting at: $99.00

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  • 2-Chloroadenosine

    2-Chloroadenosine is a metabolically stable analog of adenosine that behaves as an adenosine receptor agonist (Ki values are 300, 80 and 1900 nM for A1, A2A and A3 receptors respectively). Learn More

    Starting at: $75.00

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  • Caffeine

    Caffeine is a central nervous system stimulant, which mobilizes calcium from intracellular stores and inhibits benzodiazepine binding to GABA receptors. Learn More

    Starting at: $69.00

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  • XAC

    XAC is an adenosine receptor antagonist (IC50 values are 1.8 and 114 nM at A1 and A2 receptors respectively). Learn More

    Starting at: $95.00

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