Hydrolases
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Ceranib 1
Ceranib 1 is a ceramidase inhibitor which inhibits proliferation in SKOV3 ovarian carcinoma cells (IC50 = 3.9 μM), and induces accumulation of ceramide species and decreases sphingosine and sphingosine-1-phosphate (S1P) levels in SKOV3 cells. Learn MoreStarting at: $85.00
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PF 750
PF 750 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor that displays no activity at a range of other serine hydrolases. Learn MoreStarting at: $149.00
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SA 47
SA 47 is a selective inhibitor of fatty acid amide hydrolase (FAAH) that exhibits greater selectivity for FAAH than URB 597 against multiple carboxylesterases. Learn MoreStarting at: $109.00
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URB 597
URB 597, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, displays antiallodynic and antihyperalgesic activity in an inflammatory pain model. Learn MoreStarting at: $98.00
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SA 57
SA 57 is a potent inhibitor of fatty acid amide hydrolase (FAAH) (IC50 < 10 nM), which inhibits both human and mouse FAAH enzymes and displays inhibitory activity against FAAH, MAGL and ABHD6 in vivo. Learn MoreStarting at: $100.00
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TC-F 2
TC-F 2 is a potent, reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 values are 28 and 100 nM for human and rat FAAH respectively), which displays selectivity for FAAH over cannabinoid-related targets (IC50 > 20 μM for CB1, CB2 and TRPV1). Learn MoreStarting at: $155.00
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SC 57461A
SC 57461A is a potent and selective inhibitor of LTA4 hydrolase, which potently inhibits LTB4 production in whole blood (IC50 = 49 nM). Learn MoreStarting at: $99.00
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JW 480
JW 480 is a potent and selective inhibitor of the serine hydrolase enzyme KIAA1363 (AADACL1) (IC50 = 20 nM in mouse brain). Learn MoreStarting at: $75.00
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Flurofamide
Flurofamide is an urease inhibitor. Learn MoreStarting at: $99.00
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WWL 70
WWL 70 is a potent inhibitor of α/β-hydrolase domain 6 (ABHD6) with an IC50 of 70 nM. Learn MoreStarting at: $75.00