Androgen Receptors

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  • PF 998425

    PF 998425 is a selective non-steroidal androgen receptor (AR) antagonist (IC50 values are 26 nM and 90 nM in AR binding assays and cellular assays respectively), which displays low affinity for progesterone receptor (IC50 > 10 μM). Learn More

    Starting at: $125.00

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  • TFM-4AS-1

    TFM-4AS-1 is a potent selective androgen receptor modulator (SARM) (IC50 = 30 nM), which exhibits limited effects on reproductive tissues and sebaceous glands; does not repress AP-1-sensitive MMP-1 reporter. Learn More

    Starting at: $140.00

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  • Cl-4AS-1

    Cl-4AS-1 is a potent steroidal androgen receptor agonist (IC50 = 12 nM), which inhibits 5α-reductase type I and II (IC50 values are 6 and 10 nM respectively). Learn More

    Starting at: $140.00

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3 Item(s)

per page