M4 Receptors

PD 102807

PD 102807 is a selective M4 muscarinic receptor antagonist. IC50 values are 91, 6559, 3441, 950 and 7412 nM for human M4, M1, M2, M3, and M5 receptors respectively. Learn More

Starting at: $140.00

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VU 152100

VU 152100 is a selective positive allosteric modulator of M4 muscarinic acetylcholine receptors (mAChRs) (EC50 = 380 nM), which induces 21-fold shift in ACh potency at M4 receptor. Learn More

Starting at: $119.00

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VU 10010

VU 10010 is a selective allosteric potentiator of M4 acetylcholine receptors that binds to an allosteric site on the receptor increasing affinity for ACh and coupling to G-proteins. Learn More

Starting at: $129.00

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