κ Opioid Receptors
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nor-Binaltorphimine dihydrochloride
nor-Binaltorphimine dihydrochloride is a selective κ-opioid receptor antagonist. Learn MoreStarting at: $90.00
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(-)-U-50488 hydrochloride
(-)-U-50488 hydrochloride is a more active enantiomer of (±)-U-50488. Learn MoreStarting at: $99.00
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(+)-U-50488 hydrochloride
(+)-U-50488 hydrochloride is a less active enantiomer of (±)-U-50488. Learn MoreStarting at: $98.00
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(±)-U-50488 hydrochloride
(±)-U-50488 hydrochloride is as elective κ-opioid agonist. Learn MoreStarting at: $99.00
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GNTI dihydrochloride
GNTI dihydrochloride is a highly potent κ opioid receptor antagonist (Ki = 0.18 nM for human cloned κ receptors expressed in CHO cells), which displays 208- and 799-fold selectivity over μ and δ receptors respectively. Learn MoreStarting at: $139.00
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N-MPPP Hydrochloride
N-MPPP Hydrochloride is a high affinity κ agonist with no measured binding at μ or δ sites. Learn MoreStarting at: $110.00
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DIPPA hydrochloride
DIPPA hydrochloride is an irreversible and selective antagonist at the κ receptor, with persistent effect in vivo. Learn MoreStarting at: $100.00
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GR 89696 fumarate
Highly potent and selective κ-opioid agonist (IC50 = 0.04 nM) that may be selective for the putative κ2 receptor. Learn MoreStarting at: $135.00
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ICI 204,448 hydrochloride
ICI 204,448 hydrochloride is a peripherally acting κ agonist. Learn MoreStarting at: $95.00
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ICI 199,441 hydrochloride
ICI 199,441 hydrochloride is a highly potent κ agonist, 146-fold more active than U-50488 in vitro. Learn MoreStarting at: $95.00
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U-54494A hydrochloride
U-54494A hydrochloride is a κ-opioid agonist and anticonvulsant, which acts as an NMDA antagonist. Learn MoreStarting at: $105.00
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Salvinorin A
Salvinorin A displays high affinity at both native (Ki = 4.3 nM) and cloned (Ki = 16 nM) κ-opioid receptors. Learn MoreStarting at: $139.00