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5-HT6 Receptors
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ST 1936 oxalate
ST 1936 oxalate is a high affinity, selective agonist of 5-HT6 receptors (Ki values are 13, 168, and 245 nM for human 5-HT6, 5-HT7 and 5-HT2B receptors respectively). Learn MoreStarting at: $110.00
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EMD 386088 hydrochloride
EMD 386088 hydrochloride is a potent 5-HT6 receptor agonist (EC50 = 1.0 nM) that displays selectivity over other 5-HT receptors (IC50 values are 7.4, 110, 180, 240, 450, 620, 660 and 3000 nM for 5-HT6, 5-HT1D, 5-HT1B, 5-HT2A, 5-HT2C, 5-HT4, 5-HT1A and 5-HT7 receptors respectively). Learn MoreStarting at: $99.00
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SGS 518 oxalate
SGS 518 oxalate is a selective antagonist of the 5-HT6 subtype of the serotonin receptor. Learn MoreStarting at: $139.00
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NPS ALX Compound 4a dihydrochloride
NPS ALX Compound 4a dihydrochloride is a potent and competitive 5-HT6 antagonist (IC50 = 7.2 nM, Ki = 0.2 nM) that displays selectivity over other 5-HT and D2 receptors. Learn MoreStarting at: $139.00
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EMDT oxalate
EMDT oxalate is a selective 5-HT6 agonist (with a Ki value of 16 nM at human 5-HT6 receptors) which exhibits potency comparable to serotonin for the activation of adenylate cyclase, and displays antidepressant-like effects. Learn MoreStarting at: $119.00
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MS 245 oxalate
MS 245 oxalate is a high affinity 5-HT6 antagonist (Ki = 2.1 nM), which potentiates the hypolocomotor actions of (-)-nicotine in mice. Learn MoreStarting at: $139.00
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SB 271046 hydrochloride
SB 271046 hydrochloride is an orally active, selective 5-HT6 antagonist (pKi values are 9.02-8.92, 6.55, 6.35, 6.27, 6.05, 5.95, 5.76, 5.73, 5.62, 5.55, 5.41, 5.39, 5.27 and < 4.99 at 5-HT6, 5-HT1D, 5-HT1A, D3, 5-HT1B, 5-HT1F, α1B, 5-HT2C, 5-HT2A, D2, 5-HT2B, 5-HT7, 5-HT4 and 5-HT1E respectively) and is > 200-fold selective over 55 other receptors, enzymes and ion channels. Learn MoreStarting at: $140.00
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Ro 04-6790
Ro 04-6790 is a potent and selective 5-HT6 receptor antagonist (pKi values are 7.26 and 7.35 at rat and human 5-HT6 receptors respectively), which displays no affinity at a range of other receptors (IC50 > 10 μM). Learn MoreStarting at: $110.00
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BGC 20-761
BGC 20-761 is a selective, high affinity 5-HT6 antagonist (Ki = 20 nM). Learn MoreStarting at: $110.00
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WAY 208466 dihydrochloride
WAY 208466 dihydrochloride is a high affinity, selective 5-HT6 agonist with antidepressant and anxiolytic-like effects. Learn MoreStarting at: $149.00
