M2 Receptors
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AF-DX 116
AF-DX 116 is a selective M2 muscarinic receptor antagonist. Ki values are 64, 417, 786, 211 and 5130 nM for human recombinant M2, M1, M3, M4 and M5 muscarinic receptors, respectively. Learn MoreStarting at: $105.00
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AF-DX 384
AF-DX 384 is a potent M2/M4 selective antagonist (pKi values are 8.22, 8.00, 7.51, 7.18 and 6.27 at human M2, M4, M1, M3 and M5 receptors respectively). Learn MoreStarting at: $95.00
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(S)-(+)-Dimethindene maleate
(S)-(+)-Dimethindene maleate is an enantiomer that is a subtype-selective M2 muscarinic receptor antagonist (pKi values are 7.08, 7.78, 6.70 and 7.00 for M1, M2, M3 and M4 receptors respectively). Learn MoreStarting at: $135.00
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AQ-RA 741
AQ-RA 741 is a high affinity, selective muscarinic M2 receptor antagonist (pKi values are 8.3, 7.7 and 6.82 for M2, M1 and M3 receptors, respectively). Learn MoreStarting at: $100.00
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Arecaidine propargyl ester tosylate
Arecaidine propargyl ester tosylate is a potent muscarinic receptor agonist which shows some selectivity for cardiac versus ileal M2 receptors. Learn MoreStarting at: $70.00
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Arecaidine but-2-ynyl ester tosylate
Arecaidine but-2-ynyl ester tosylate is a potent muscarinic agonist, 4.6-fold selective for M2 receptors in the atrium versus those in the ileum. Learn MoreStarting at: $95.00