CB2 Receptors

11 Item(s)

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  • SER 601

    SER 601 is a potent and selective CB2 receptor agonist (Ki values are 6.3 nM and 1.2 μM for CB2 and CB1 receptors respectively). Learn More

    Starting at: $109.00

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  • CB 65

    CB 65 is a high affinity and selective CB2 receptor agonist. Learn More

    Starting at: $139.00

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  • GP 1a

    GP 1a is a highly selective CB2 receptor agonist that increases P-ERK1/2 expression in HL-60 cells in vitro with Ki values are 0.037 and 363 nM for CB2 and CB1 receptors respectively. Learn More

    Starting at: $150.00

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  • AM 630

    Immepip dihydrobromide is a potent histamine H3 receptor agonist which also binds to H4 receptors (Ki values are 0.4 and 9 nM at human recombinant H3 and H4 receptors respectively). Learn More

    Starting at: $135.00

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  • JTE 907

    JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist, which binds with high affinity to rat, mouse and human CB2 receptors (Ki values are 0.38, 1.55 and 35.9 nM respectively). Learn More

    Starting at: $139.00

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  • HU 308

    HU 308 is a potent and selective CB2 receptor agonist (Ki values are 22.7 nM and > 10 μM for CB2 and CB1 receptors respectively, EC50 = 5.57 nM) which displays antiallodynic activity in the rat hindpaw incision model of postoperative pain. Learn More

    Starting at: $179.00

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  • GW 405833

    GW 405833 is a potent and selective CB2 receptor partial agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%) which binds with high affinity to both human and rat CB2 receptors and displays ~ 1200-fold selectivity over CB1 (Ki values are 3.92 and 4772 nM for human recombinant CB2 and CB1 receptors respectively). Learn More

    Starting at: $135.00

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  • L-759,656

    Highly selective CB2 receptor agonist (Ki values are 11.8 and 4888 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 3.1 nM). Learn More

    Starting at: $180.00

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  • L-759,633

    L-759,633 is a high affinity, selective CB2 receptor agonist (Ki values are 6.4 and 1043 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 8.1 nM). Learn More

    Starting at: $180.00

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  • JWH 015

    JWH 015 is a selective CB2 agonist (Ki values are 13.8 and 383 nM as measured at human cloned CB2 and CB1 receptors expressed in CHO cells). Learn More

    Starting at: $50.00

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  • GP 2a

    GP 2a is a selective CB2 receptor agonist with Ki values of 7.6 and 900 nM for CB2 and CB1 receptors respectively. Learn More

    Starting at: $169.00

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11 Item(s)

per page