CB2 Receptors
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SER 601
SER 601 is a potent and selective CB2 receptor agonist (Ki values are 6.3 nM and 1.2 μM for CB2 and CB1 receptors respectively). Learn MoreStarting at: $109.00
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CB 65
CB 65 is a high affinity and selective CB2 receptor agonist. Learn MoreStarting at: $139.00
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GP 1a
GP 1a is a highly selective CB2 receptor agonist that increases P-ERK1/2 expression in HL-60 cells in vitro with Ki values are 0.037 and 363 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $150.00
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AM 630
Immepip dihydrobromide is a potent histamine H3 receptor agonist which also binds to H4 receptors (Ki values are 0.4 and 9 nM at human recombinant H3 and H4 receptors respectively). Learn MoreStarting at: $135.00
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JTE 907
JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist, which binds with high affinity to rat, mouse and human CB2 receptors (Ki values are 0.38, 1.55 and 35.9 nM respectively). Learn MoreStarting at: $139.00
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HU 308
HU 308 is a potent and selective CB2 receptor agonist (Ki values are 22.7 nM and > 10 μM for CB2 and CB1 receptors respectively, EC50 = 5.57 nM) which displays antiallodynic activity in the rat hindpaw incision model of postoperative pain. Learn MoreStarting at: $179.00
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GW 405833
GW 405833 is a potent and selective CB2 receptor partial agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%) which binds with high affinity to both human and rat CB2 receptors and displays ~ 1200-fold selectivity over CB1 (Ki values are 3.92 and 4772 nM for human recombinant CB2 and CB1 receptors respectively). Learn MoreStarting at: $135.00
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L-759,656
Highly selective CB2 receptor agonist (Ki values are 11.8 and 4888 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 3.1 nM). Learn MoreStarting at: $180.00
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L-759,633
L-759,633 is a high affinity, selective CB2 receptor agonist (Ki values are 6.4 and 1043 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 8.1 nM). Learn MoreStarting at: $180.00
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JWH 015
JWH 015 is a selective CB2 agonist (Ki values are 13.8 and 383 nM as measured at human cloned CB2 and CB1 receptors expressed in CHO cells). Learn MoreStarting at: $50.00
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GP 2a
GP 2a is a selective CB2 receptor agonist with Ki values of 7.6 and 900 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $169.00