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Enzymes
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ARL 67156 trisodium salt
NU 2058 is a cyclin-dependent kinase (cdk) 1 and cdk2 inhibitor (Ki values are 5 and 12 μM respectively), which inhibits growth of human tumor cells in vitro (mean GI50 = 13 μM) and DNA topoisomerase II ATPase activity (IC50 = 300 μM). Learn MoreStarting at: $155.00
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Tacrine hydrochloride
AIDA is a relatively potent and selective antagonist of group I metabotropic glutamate receptors (mGlu1a), having no effect on group II (mGlu2) or group III (mGlu4) receptors expressed individually in baby hamster kidney cells. Learn MoreStarting at: $60.00
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Ambenonium dichloride
Ambenonium dichloride is a extremely potent, selective and rapidly reversible inhibitor of acetylcholinesterase (AChE) with IC50 values =0.000698 and 8.20 μM at AChE and BChE respectively. Learn MoreStarting at: $99.00
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Physostigmine hemisulfate
Physostigmine hemisulfate is a cholinesterase inhibitor. Learn MoreStarting at: $33.00
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PSB 069
PSB 069 is a non-selective nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitor. Learn MoreStarting at: $109.00
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CI 898 trihydrochloride
CI 898 trihydrochloride is a potent lipophilic inhibitor of dihydrofolate reductase (DHFR) that inhibits protozoal, bacterial and human DHFR with IC50 values of 1.4, 6.1 and 3.2 nM respectively. Learn MoreStarting at: $139.00
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PI 828
PI 828 is a PI 3-Kinase inhibitor with IC50 values of 0.098, 0.183, 0.227 and 1.967 μM for p110β, p110α, p110δ and p110γ respectively. Learn MoreStarting at: $69.00
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Alda 1
Alda 1 is an activator of aldehyde dehydrogenase 2 (ALDH2). Increases activity of wild-type ALDH2*1 and variant ALDH2*2 (by ~2-fold and 11-fold respectively). Learn MoreStarting at: $59.00
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Acephate
Anticholinesterase insecticide that produces cholinotoxicity, which displays weak inhibition of rat acetylcholinesterase (AChE) but potently inhibits cockroach AChE. Learn MoreStarting at: $59.00
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Fumagillin
Fumagillin is an antibiotic and antiangiogenic agent, which covalently binds and inhibits methionine aminopeptidase-2. Learn MoreStarting at: $119.00
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Galanthamine hydrobromide
Galanthamine hydrobromide is a long-acting, centrally active acetylcholinesterase inhibitor (IC50 = 410 nM) and allosteric potentiator at neuronal nicotinic ACh receptors. Learn MoreStarting at: $75.00
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Phenserine
Phenserine is a Physostigmine analog that inhibits acetylcholinesterase.Phenserin also inhibits production of amyloid precursor protein (APP) and A&beta and improves morris water maze performance of scopolamine-treated rats. Learn MoreStarting at: $95.00
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PF 04691502
PF 04691502 is an potent and selective dual ATP-competitive PI 3-K/mTOR inhibitor (Ki values are 1.6, 1.8, 1.9, 2.1 and 16 nM for human PI 3-K δ, α, γ, β, and mTOR, respectively). Learn MoreStarting at: $145.00
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PSB 06126
PSB 06126 is a nucleoside triphosphate diphosphohydrolase 3 (NTPDase 3) inhibitor, which inhibits rat NTPDase 3 at low micromolar concentrations and display selectivity over NTPDase 1 and NTPDase 2. Learn MoreStarting at: $120.00
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PE 154
PE 154 is a potent fluorescent inhibitor of human acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) (IC50 values are 280 pM and 16 nM respectively), which targets and labels β-amyloid plaques in histochemical analysis. Learn MoreStarting at: $160.00
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Rivastigmine tartrate
Rivastigmine tartrate is a dual cholinesterase inhibitor (ChEI) which inhibits both butyrylcholinesterase (BChE) and acetylcholinesterase (AChE). Learn MoreStarting at: $70.00
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Tin protoporphyrin IX dichloride
Tin protoporphyrin IX dichloride is a potent inhibitor of heme oxygenase which prevents hyperbilirubinemia in neonates. Learn MoreStarting at: $85.00
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WIN 18446
WIN 18446 is an inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2) (IC50 = 0.3 μM) which inhibits the biosynthesis of retinoic acid from retinol in neonatal and adult murine testis. Learn MoreStarting at: $80.00
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LY 303511
LY 303511 is a negative control compound with respect to LY 294002 PI 3-kinase inhibitory activity which blocks voltage-gated potassium (Kv) channels (IC50 = 64.6 μM) and inhibits IL-1β-stimulated NF-κB activation, attenuating MCP-1 expression. Antiproliferative. Learn MoreStarting at: $75.00
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CMPD-1
CMPD-1 is a non-ATP-competitive, selective inhibitor of p38α-mediated MK2a (mitogen-activated protein kinase-activated protein kinase 2a) phosphorylation (apparent Ki = 330 nM). Does not inhibit p38α-mediated phosphorylation of the two other known p38 substrates, MBP and ATF-2. Learn MoreStarting at: $119.00
