Glycogen Synthase Kinase 3

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  • TCS 2002

    TCS 2002 is a potent inhibitor of GSK-3β (IC50 = 35 nM), that inhibits cold water stress-induced tau hyperphosphorylation in the mouse brain. Learn More

    Starting at: $129.00

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  • TC-G 24

    TC-G 24 is a potent GSK-3β inhibitor (IC50 = 17 nM), which displays selectivity for GSK-3β over CDK2 (22% inhibition at 10 μM). Learn More

    Starting at: $135.00

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  • A 1070722

    A 1070722 is a potent glycogen synthase kinase-3 (GSK-3) inhibitor (Ki = 0.6 nM for GSK-3α and GSK-3β) which displays high selectivity (> 50-fold) for GSK-3 over a panel of other kinases tested, including CDK family members. Learn More

    Starting at: $135.00

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  • 3F8

    L-755,507 is a potent β3-adrenergic receptor partial agonist > 1000-fold selective over β1- and β2-adrenoceptors (EC50 values are 0.43, 580 and > 10000 nM for activation of cloned human β3-, β1- and β2-adrenoceptors respectively). Learn More

    Starting at: $115.00

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  • Indirubin-3'-oxime

    ARL 67156 trisodium salt is a selective ecto-ATPase inhibitor (pIC50 = 4.62 and 5.1 in human blood and rat vas deferens respectively). Learn More

    Starting at: $110.00

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  • BIO

    BIO is a potent and selective, ATP-competitive glycogen synthase kinase-3 (GSK-3) inhibitor that maintains self-renewal and pluripotency in embryonic stem cells via activation of the Wnt signaling pathway in vitro and also promotes proliferation and dedifferentiation in cardiomyocytes. Learn More

    Starting at: $109.00

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  • BIO-acetoxime

    BIO-acetoxime is a selective GSK-3α/β inhibitor that induces Wnt signaling and inhibits CD8+ T cell effector differentiation. Learn More

    Starting at: $89.00

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  • MeBIO

    MeBIO is an Aryl hydrocarbon receptor (AhR) agonist that causes redistribution of AhR to the nucleus. Learn More

    Starting at: $119.00

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  • PF 04885614

    PF 04885614 is a potent NaV1.8 inhibitor (IC50 = 53 nM for human NaV1.8 channel), which exhibits selectivity for hNaV1.8 over hNaV1.6, hNaV1.7, hNaV1.1, hNaV1.2 and hNaV1.5 (IC50 values are 4.2, 7.0, 11, 16 and 27 μM respectively). Learn More

    Starting at: $125.00

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9 Item(s)

per page