Src Kinase
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KB SRC 4
KB SRC 4 is a potent and selective c-Src inhibitor (Ki = 44 nM) and significantly inhibits cell growth in 4T1 mammary carcinoma tumor cells. Learn MoreStarting at: $175.00
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MNS
MNS is a selective inhibitor of Src and Syk tyrosine kinases which displays antiaggregative activity via inhibition of GPIIb/IIIa activation (IC50 = 12.7 μM for thrombin-induced platelet aggregation). Learn MoreStarting at: $65.00
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Src I1
Src I1 is a potent, competitive dual site (ATP- and peptide-binding) Src kinase inhibitor (IC50 values are 44 and 88 nM for Src and Lck respectively) which inhibits VEGFR2 and c-fms at higher concentrations (IC50 values are 0.32 and 30 μM respectively). Learn MoreStarting at: $120.00
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AZM 475271
AZM 475271 is a src tyrosine kinase inhibitor, which reduces tumor size, vascularity and metastasis, and increases apoptosis in human pancreatic cells grown in nude mice. Learn MoreStarting at: $179.00
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Damnacanthal
Damnacanthal is a potent inhibitor of p56lck tyrosine kinase activity (IC50 = 17 nM for inhibition of autophosphorylation), which displays 7- to 20-fold selectivity over p59fyn and p60src tyrosine kinases, > 40-fold selectivity over c-ErbB2, EGF- and insulin-receptor tyrosine kinases, and > 100-fold selectivity over PKA and PKC. Learn MoreStarting at: $115.00
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PP 3
PP 3 is a negative control for the Src kinase inhibitor PP 2 Inhibits EGFR kinase (IC50 = 2.7 μM). Learn MoreStarting at: $139.00
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Herbimycin A
Herbimycin A is an ansamycin antibiotic that acts as a Src family kinase inhibitor that binds to the SH domain and inhibits the activity of p60v-src and p210BCR-ABL. Learn MoreStarting at: $125.00