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5-HT Receptors
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NPEC-caged-serotonin
NPEC-caged-serotonin is a NPEC ((N)-1-(2-nitrophenyl)ethyl) caged version of serotonin. Learn MoreStarting at: $135.00
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Methiothepin maleate
Methiothepin maleate is a potent 5-HT2 antagonist, also active as 5-HT1 antagonist, which displays affinity for rodent 5-HT5B, 5-HT5A, 5-HT7 and 5-HT6 receptors (pK1 values are 6.6, 7.0, 8.4 and 8.7 respectively). Learn MoreStarting at: $65.00
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Serotonin hydrochloride
Serotonin hydrochloride is an Endogenous agonist at 5-HT receptors and endogenous substrate for 5-HT transporters. Learn MoreStarting at: $60.00
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LY 215840
LY 215840 is a 5-HT2/5-HT7 receptor antagonist which reduces stimulatory effect of serotonin on aldosterone secretion and 5-HT-induced cAMP formation (pKB = 8.26). Learn MoreStarting at: $135.00
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Methysergide maleate
Methysergide maleate is a mixed 5-HT1/5-HT2 receptor antagonist. Learn MoreStarting at: $115.00
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Methylergometrine maleate
Methylergometrine maleate is an active metabolite of methysergide. Learn MoreStarting at: $80.00
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Psilocin
PsilocinNon, an active metabolite of psilocybinm, is a selective serotonin receptor agonist. Active metabolite of psilocybin. Learn MoreStarting at: $219.00
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AS 19
AS 19 is a potent 5-HT7 receptor agonist (IC50 = 0.83 nM), that enhances memory consolidation and reverses scopolamine- or dizocilpine-induced amnesia in vivo. Learn MoreStarting at: $109.00
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LP 44
LP 44 is a high affinity 5-HT7 receptor agonist that displays selectivity over 5-HT1A and 5-HT2A receptors (200- and > 1000-fold respectively). Learn MoreStarting at: $145.00
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LP 12 hydrochloride
LP 12 hydrochloride is a 5-HT7 receptor agonist displaying selectivity over D2, 5-HT1A and 5-HT2A receptors (Ki values are 0.22, 7.3, 52.7 and 326 nM respectively), which induces relaxation of substance P-induced contractions in guinea pig ileum (EC50 = 1.77 μM). Learn MoreStarting at: $135.00
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LP 20 hydrochloride
LP 20 hydrochloride is a ligand of the 5-HT7 receptor (Ki = 2.6 nM) which exhibits agonist and antagonist activity. It also displays selectivity over adrenergic α1 and 5-HT1A receptors (Ki values are 156 and 476 nM respectively). Learn MoreStarting at: $115.00
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SB 258719 hydrochloride
SB 258719 hydrochloride is a selective 5-HT7 receptor antagonist that displays > 100-fold selectivity over a range of other receptors. Learn MoreStarting at: $119.00
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SB 269970 hydrochloride
SB 269970 hydrochloride is a potent and selective 5-HT7 receptor antagonist (pKi values are 8.9, 7.2 and 6.0 for 5-HT7A, 5-HT5A and 5-HT1B and < 6.0 for 5-HT1A, 5-HT1D, 5-HT1E, 5-HT1F, 5-HT2A, 5-HT2B, 5-HT2C, 5-HT4 and 5-HT6 receptors respectively). Learn MoreStarting at: $135.00
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5-Carboxamidotryptamine maleate
5-Carboxamidotryptamine maleate is a 5-HT1 agonist with high affinity at 5-HT1A, 5-HT1B , 5-HT1D, 5-ht5 and 5-HT7 receptors. Learn MoreStarting at: $139.00
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ST 1936 oxalate
ST 1936 oxalate is a high affinity, selective agonist of 5-HT6 receptors (Ki values are 13, 168, and 245 nM for human 5-HT6, 5-HT7 and 5-HT2B receptors respectively). Learn MoreStarting at: $110.00
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BGC 20-761
BGC 20-761 is a selective, high affinity 5-HT6 antagonist (Ki = 20 nM). Learn MoreStarting at: $110.00
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Ro 04-6790
Ro 04-6790 is a potent and selective 5-HT6 receptor antagonist (pKi values are 7.26 and 7.35 at rat and human 5-HT6 receptors respectively), which displays no affinity at a range of other receptors (IC50 > 10 μM). Learn MoreStarting at: $110.00
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SB 271046 hydrochloride
SB 271046 hydrochloride is an orally active, selective 5-HT6 antagonist (pKi values are 9.02-8.92, 6.55, 6.35, 6.27, 6.05, 5.95, 5.76, 5.73, 5.62, 5.55, 5.41, 5.39, 5.27 and < 4.99 at 5-HT6, 5-HT1D, 5-HT1A, D3, 5-HT1B, 5-HT1F, α1B, 5-HT2C, 5-HT2A, D2, 5-HT2B, 5-HT7, 5-HT4 and 5-HT1E respectively) and is > 200-fold selective over 55 other receptors, enzymes and ion channels. Learn MoreStarting at: $140.00
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MS 245 oxalate
MS 245 oxalate is a high affinity 5-HT6 antagonist (Ki = 2.1 nM), which potentiates the hypolocomotor actions of (-)-nicotine in mice. Learn MoreStarting at: $139.00
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EMDT oxalate
EMDT oxalate is a selective 5-HT6 agonist (with a Ki value of 16 nM at human 5-HT6 receptors) which exhibits potency comparable to serotonin for the activation of adenylate cyclase, and displays antidepressant-like effects. Learn MoreStarting at: $119.00
