7-TM Receptors

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  • Pronethalol hydrochloride

    Pronethalol hydrochloride is a ??-adrenergic antagonist, clinically effective in the treatment of angina pectoris and some arrhythmias. Learn More

    Starting at: $69.00

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  • CY 208-243

    CY 208-243 is a centrally active dopamine D1 receptor agonist, selective over D2 receptor sites, which stimulates adenylate cyclase in rat striatal homogenates with an EC50 of 125 nM, that exerts antiParkinsonian activity in animal models. Learn More

    Starting at: $139.00

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  • DPCPX

    DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Learn More

    Starting at: $119.00

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  • Z-Cyclopentyl-AP4

    Z-Cyclopentyl-AP4 is a group III mGlu receptor agonist that exhibits higher potency at mGlu4 than mGlu8 (EC50 values are 49 and 124 μM respectively) with no activity at mGlu7. And selectively inhibits synaptic activity in the lateral perforant pathway (IC50 values are 130 and 1859 μM in the lateral and medial perforant pathways respectively). Learn More

    Starting at: $129.00

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  • (±)-5'-Chloro-5'-deoxy-ENBA

    (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist (Ki values are 0.51, 1290, 1340 and 2740 nM at A1, A3, A2A and A2B receptors respectively). Learn More

    Starting at: $135.00

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  • SKF 77434 hydrobromide

    SKF 77434 hydrobromide is a selective dopamine D1-like receptor partial agonist (IC50 values are 19.7 and 2425 nM for binding to D1-like and D2-like receptors respectively). Learn More

    Starting at: $79.00

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  • Cevimeline hydrochloride

    Cevimeline hydrochloride is a selective M1 receptor agonist which induces atropine-sensitive contractions of isolated guinea pig ilea and trachea preparations (EC50 values are 3.5 and 3 μM respectively). Learn More

    Starting at: $95.00

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  • VU 0155041

    VU 0155041 is a potent, positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50 = 798 and 693 nM at human and rat mGlu4 receptors respectively). Learn More

    Starting at: $120.00

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  • Naltrindole hydrochloride

    Naltrindole hydrochloride is a highly selective non-peptide δ opioid antagonist, showing 223- and 346-fold greater activity at δ than at μ and κ opioid receptors. Learn More

    Starting at: $95.00

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  • Naltriben mesylate

    Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively), which displays selectivity for the δ2 subtype in vivo. Learn More

    Starting at: $100.00

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  • VU 0357017 hydrochloride

    VU 0357017 hydrochloride is a positive allosteric modulator of muscarinic M1 receptors (EC50 = 198 nM), which displays no activity at M2-M5 at concentrations up to 30 μM. Learn More

    Starting at: $110.00

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  • VU 0255035

    VU 0255035 is a highly selective muscarinic M1 antagonist (Ki = 14.87 nM), which targets the M1 orthosteric site and reduces pilocarpine-induced seizures in mice. Learn More

    Starting at: $110.00

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  • Tocrifluor T1117

    Tocrifluor T1117 is a novel fluorescent form of AM 251, which conjugated with 5-carboxytetramethylrhodamine (5-TAMRA) that fluoresces at 543nm excitation (590nm emission), and displays GPR55 binding activity. Learn More

    Starting at: $200.00

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  • N-Benzylnaltrindole hydrochloride

    N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist with a long duration of action in vivo. Learn More

    Starting at: $95.00

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  • (RS)-PPG

    (RS)-PPG is a potent and selective group III metabotropic glutamate receptor agonist, with approximately 25-fold preference for hmGlu8. Learn More

    Starting at: $100.00

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  • Dihydrexidine hydrochloride

    Dihydrexidine hydrochloride is a potent, full efficacy dopamine D1 agonist which shows no agonist activity at peripheral D2 receptors or adrenoceptors at doses which cause maximal stimulation of D1 sites. Learn More

    Starting at: $95.00

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  • GR 79236

    GR 79236 is a adenosine A1 receptor agonist (Ki = 3.1 nM). Learn More

    Starting at: $155.00

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  • TCN 238

    TCN 238 is a positive allosteric modulator of mGlu4 receptors (EC50 = 1.0 μM for human and rat mGlu4 receptors). Learn More

    Starting at: $105.00

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  • NPEC-caged-(S)-3,4-DCPG

    NPEC-caged-(S)-3,4-DCPG is a (S)-3,4-DCPG caged with the photosensitive 1-(2-nitrophenyl)ethoxycarbonyl group. Learn More

    Starting at: $215.00

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  • VU 0155041 sodium salt

    VU 0155041 sodium salt is a potent, positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50 = 798 and 693 nM at human and rat mGlu4 receptors respectively). Learn More

    Starting at: $50.00

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