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7-TM Receptors
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ACPA
ACPA is a potent and selective CB1 agonist (Ki = 2.2 nM) which displays 325-fold selectivity over CB2 receptors. Learn MoreStarting at: $69.00
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O-Phospho-L-serine
O-Phospho-L-serine is a group III metabotropic glutamate receptor agonist; analog of L-AP4, which inhibits proliferation and enhances neuronal differentiation in progenitor cells. Learn MoreStarting at: $59.00
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N6-Cyclopentyladenosine
N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 2.3, 790 and 43 nM for human A1, A2A and A3 receptors respectively; EC50 = 18600 nM for hA2B). Learn MoreStarting at: $89.00
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MMPIP hydrochloride
MMPIP hydrochloride is a potent allosteric mGlu7-selective receptor antagonist, which inhibits agonist-induced intracellular calcium mobilization and cAMP accumulation (IC50 values are 26 and 610 nM). Learn MoreStarting at: $65.00
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NIDA 41020
NIDA 41020 is a high affinity CB1 receptor antagonist (Ki = 4.1 nM), which exhibits significantly reduced lipophilicity compared to other CB1 antagonists. Learn MoreStarting at: $139.00
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(R)-(+)-Propranolol hydrochloride
(R)-(+)-Propranolol hydrochloride is a less active enantiomer of the β-adrenoceptor antagonist propranolol. Learn MoreStarting at: $69.00
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Terfenadine
Terfenadine is a histamine H1 receptor antagonist, which also blocks KV11.1 (hERG) and Kir6 (KATP) channels (IC50 values are 204 nM and 1.2 μM respectively). Learn MoreStarting at: $49.00
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Doxepin hydrochloride
BMS 453 is a synthetic retinoid. Retinoic acid receptor β (RARβ) agonist in vivo; RARα and RARγ antagonist in vitro. Learn MoreStarting at: $55.00
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MPPG
MTPG is a group II/group III metabotropic glutamate receptor antagonist, showing selectivity for group II in electrophysiological studies. Learn MoreStarting at: $135.00
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PSB 36
PSB 36 is a Potent and selective A1 adenosine receptor antagonist with binding affinities of 0.12, 187, 552, 6500 and 2300 nM for rA1, hA2B, rA2A, rA3 and hA3 receptors respectively. Learn MoreStarting at: $129.00
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ICI 89406
ICI 89406 is a β-adrenergic antagonist and low efficacy partial agonist. Learn MoreStarting at: $91.00
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SDZ 21009
SDZ 21009 is a β-adrenoceptor and 5-HT1A/1B receptor antagonist. pKB/pA2 values are 8.3 and 8.0 for 5-HT1A and 5-HT1B receptors respectively. Learn MoreStarting at: $135.00
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2-Chloro-N6-cyclopentyladenosine
2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 0.8, 2300 and 42 nM for human A1, A2A and A3 receptors respectively; EC50 = 18800 nM for hA2B). Learn MoreStarting at: $99.00
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L-AP4
L-AP4 is a selective group III metabotropic glutamate receptor agonist. Synaptic depressant. Agonist at the quisqualate-sensitized AP6 site in hippocampus. Learn MoreStarting at: $60.00
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SLV 320
SLV 320 is a potent and selective adenosine A1 receptor antagonist (Ki values are 1, 200, 398 and 3981 nM at human A1, A3, A2A and A2B receptors respectively). Learn MoreStarting at: $105.00
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LE 300
LE 300 is a potent and selective dopamine D1 receptor antagonist (Ki values are 0.08 - 1.9 nM and 6 - 45 nM for D1 and D2 receptors respectively), which also displays moderate affinity for the 5-HT2A receptor (Ki = 20 nM). Active in vivo. Learn MoreStarting at: $139.00
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Pirenzepine dihydrochloride
Pirenzepine dihydrochloride is a M1 muscarinic receptor selective antagonist. Learn MoreStarting at: $65.00
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Oleamide
Oleamide endogenous sleep-inducing lipid, which acts as an agonist at the CB1 cannabinoid receptor (EC50 = 1.64 μM). Learn MoreStarting at: $59.00
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2-Pyridylethylamine dihydrochloride
2-Pyridylethylamine dihydrochloride is a histamine H1 receptor agonist that produces vasoconstriction in vivo. Learn MoreStarting at: $69.00
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UBP1112
UBP1112 is a selective group III mGlu receptor antagonist (apparent Kd values are 5.1 and 488 μM for group III and group II mGlu receptors respectively; IC50 > 1 mM for group I, NMDA, AMPA and kainate receptors). Learn MoreStarting at: $139.00
