5-HT1A Receptors
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Cyanopindolol hemifumarate
Cyanopindolol hemifumarate is a 5-HT1A/1B antagonist with roughly equal affinity at each receptor; also a β-adrenoceptor antagonist. Learn MoreStarting at: $99.00
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Xaliproden hydrochloride
Xaliproden hydrochloride is an orally active, full agonist at 5-HT1A receptors that is > 300-fold selective over other 5-HT receptor subtypes with an IC50 value of > 650 nM. Learn MoreStarting at: $105.00
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BP 554 maleate
BP 554 maleate is a selective 5-HT1A agonist. Learn MoreStarting at: $95.00
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(R)-(+)-8-Hydroxy-DPAT hydrobromide
(R)-(+)-8-Hydroxy-DPAT hydrobromide is a full 5-HT1A serotonin receptor agonist that reduces hippocampal 5-HT levels following systemic administration in rats in vivo. It is more active enantiomer of 8-Hydroxy-DPAT hydrobromide. Learn MoreStarting at: $109.00
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8-Hydroxy-DPAT hydrobromide
8-Hydroxy-DPAT hydrobromide is a standard selective 5-HT1A agonist that reduces hippocampal 5-HT levels following systemic administration in rats in vivo. Learn MoreStarting at: $59.00
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WAY 100635 maleate
WAY 100635 maleate is a potent, silent antagonist of 5-HT1A receptors with 100-fold selectivity for 5-HT1A over other 5-HT subtypes. It also has agonist activity at dopamine D4 receptors. Learn MoreStarting at: $119.00
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8-Hydroxy-PIPAT oxalate
SCH 58261 is a potent and selective A2A adenosine receptor competitive antagonist (Ki = 1.3 nM). Displays 323-, 53- and 100-fold selectivity over A1, A2B and A3 receptors, respectively. Learn MoreStarting at: $120.00
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MM 77 dihydrochloride
This ligand has uniquely high affinity and selectivity for the D3 receptor. Learn MoreStarting at: $95.00
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Buspirone hydrochloride
Buspirone hydrochloride is a classic 5-HT1A partial agonist with relatively high affinity (Ki = 9.3 - 29.5 nM). Learn MoreStarting at: $49.00
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(S)-WAY 100135 dihydrochloride
(S)-WAY 100135 dihydrochloride is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM). Learn MoreStarting at: $110.00
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S 14506 hydrochloride
S 14506 hydrochloride is a highly potent selective 5-HT1A receptor full agonist (pKi values are 9.0, 6.6, 7.5, 6.6 and < 6.0 for 5-HT1A, 5-HT1B, 5-HT1C, 5-HT2 and 5-HT3 receptors respectively). Learn MoreStarting at: $135.00
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MDL 73005EF hydrochloride
MDL 73005EF hydrochloride is a potent and selective 5-HT1A receptor antagonist, which has partial agonist properties. Learn MoreStarting at: $90.00
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MDL 72832 hydrochloride
MDL 72832 hydrochloride is a potent ligand at 5-HT1A receptors, with mixed agonist and antagonist properties. Learn MoreStarting at: $90.00
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Ipsapirone
Ipsapirone is a selective 5-HT1A receptor agonist with a Ki value of 10 nM. Learn MoreStarting at: $99.00