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Kinases
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(5Z)-7-Oxozeaenol
(5Z)-7-Oxozeaenol is a resorcyclic lactone of fungal origin that acts as a potent and selective transforming growth factor-β-activated kinase 1 (TAK1) mitogen-activated protein kinase kinase kinase (MAPKKK) inhibitor (IC50 = 8 nM). Learn MoreStarting at: $109.00
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PIR 3.5
PIR 3.5 is a non-competitive inhibitor of group I p21-activated kinase (Pak1). Learn MoreStarting at: $92.00
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TNP
TNP is a Reversible inositol hexakisphosphate kinase (IP6K) inhibitor with IC50 = 0.47 μM for inhibition of InsP7 formation. Learn MoreStarting at: $139.00
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Harmine
Harmine is a potent and selective inhibitor of Dyrk1A (IC50 values are 80, 800 and 900 nM for Dyrk1A, Dyrk3 and Dyrk2 respectively), which shown to inhibit direct phosphorylation of tau by Dyrk1A (IC50 = 700 nM). Learn MoreStarting at: $49.00
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DCA
DCA is an inhibitor of mitochondrial pyruvate dehydrogenase kinase (PDK), which shifts pyruvate metabolism from glycolysis and lactate production to glucose oxidation in the mitochondria, and induces mitochondrial-dependent apoptosis and reverses the inhibition/downregulation of KV1.5 channels in cancer but not normal cells. Learn MoreStarting at: $55.00
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PF 06465469
PF 06465469 is a potent inhibitor of interleukin-2 inducible T cell kinase (ITK) (IC50 = 2 nM)which exhibits inhibitory activity against Bruton's tyrosine kinase (BTK) (IC50 = 2 nM). Learn MoreStarting at: $180.00
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KH CB19
KH CB19 is a selective, potent inhibitor of CDC2-like kinase (CLK) 1 and 4 (IC50 = 20 nM for CLK1) which suppresses serine/arginine-rich protein phosphorylation by CLKs under proinflammatory conditions, and displays selectivity over a panel of 71 protein kinases. Learn MoreStarting at: $65.00
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Ro 31-8220 mesylate
Ro 31-8220 mesylate is a protein kinase C inhibitor, with activity at other protein kinases (IC50 values are 33, 3, 8, 15 and 38 nM for PKCα, MAPKAP-K1b, MSK1, GSK3β and S6K1 respectively). Learn MoreStarting at: $95.00
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H-9 dihydrochloride
H-9 dihydrochloride is a protein kinase inhibitor that inhibits PKA, PKG, CaMK II, PKC, casein kinase I and casein kinase II. Learn MoreStarting at: $89.00
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H-7 dihydrochloride
H-7 dihydrochloride is a protein kinase inhibitor. Learn MoreStarting at: $95.00
