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Enzymes
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MMPX
MMPX is a specific inhibitor of calmodulin-sensitive cyclic GMP phosphodiesterase. Learn MoreStarting at: $119.00
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Enoximone
Enoximone is increases intracellular cyclic AMP (cAMP) concentrations and enhances myocardial contractility. Learn MoreStarting at: $119.00
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BC 11-38
BC 11-38 is a selective phosphodiesterase (PDE) 11 inhibitor that elevates cAMP levels and cortisol production in H295R human adenocarcinoma cells. Learn MoreStarting at: $129.00
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CDP 840 hydrochloride
(S)-3,5-DHPG is a selective group I mGlu receptor agonist. Learn MoreStarting at: $135.00
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Etazolate hydrochloride
Etazolate hydrochloride is a phosphodiesterase inhibitor, selective for PDE4 (IC50 = 2.0 μM). Learn MoreStarting at: $79.00
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BRL 50481
BRL 50481 is a selective, substrate-competitive inhibitor of phosphodiesterase (PDE) 7 (Ki = 180 nM), which displays > 200-fold selectivity over PDE1B, PDE1C, PDE2, PDE3, PDE4A4 and PDE5. Learn MoreStarting at: $89.00
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TBB
TBB is a cell-permeable, selective inhibitor of casein kinase-2 (CK2) (IC50 = 0.9 and 1.6 μM for rat liver and human recombinant CK2 respectively). Learn MoreStarting at: $65.00
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(R)-DRF053 dihydrochloride
(R)-DRF053 dihydrochloride is a potent, ATP-competitive inhibitor of cyclin-dependent kinase (cdk) and casein kinase 1 (CK1) (IC50 values are 220, 80 and 14 nM for cdk1/cyclin B, cdk5/p25 and CK1 respectively), which also shown to inhibit amyloid-β production in N2A-APP695 cells. Learn MoreStarting at: $140.00
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PF 4800567 hydrochloride
PF 4800567 hydrochloride is a selective casein kinase 1ε inhibitor; displays 22-fold greater potency towards CK1ε than CK1δ (IC50 values are 32 and 711 nM for CK1ε and CK1δ respectively). Learn MoreStarting at: $125.00
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(-)-Terreic acid
Selective inhibitor of Bruton's tyrosine kinase (BTK), which inhibits the interaction between PKCbII and BTK (IC50 ~ 30 mM) and the catalytic activity of BTK but does not affect the activity of PKC. Learn MoreStarting at: $155.00
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Y-29794 oxalate
Y-29794 oxalate is an inhibitor of prolyl endopeptidase, a serine peptidase that may be implicated in the biosynthesis of amyloid β-peptide. Learn MoreStarting at: $140.00
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Butabindide oxalate
Butabindide oxalate is a potent, reversible, selective and competitive inhibitor of a CCK-inactivating serine protease (tripeptidyl peptidase II) (Ki = 7 nM). Learn MoreStarting at: $135.00
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CGS 35066
CGS 35066 is a potent endothelin-converting enzyme (ECE) inhibitor that displays > 100-fold selectivity over neutral endopeptidase 24.11 (IC50 values are 22 and 2300 nM respectively). Learn MoreStarting at: $179.00
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LFM-A13
LFM-A13 is a potent and selective inhibitor of Bruton's tyrosine kinase (BTK) that inhibits recombinant BTK with an IC50 value of 2.5 μM and has no activity on other protein kinases. Learn MoreStarting at: $129.00
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UAMC 00039 dihydrochloride
UAMC 00039 dihydrochloride is potent inhibitor of dipeptidyl peptidase II (DPP-II) with selectivity for DPP-II against DPP-9, DPP-8 and DPP-IV. Learn MoreStarting at: $169.00
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Cilastatin sodium
Cilastatin sodium is a dipeptidase inhibitor that inhibits metabolism of LTD4 to LTE4 and the hydrolysis of β-lactam antibiotics. Learn MoreStarting at: $89.00
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Nafamostat mesylate
Nafamostat mesylate is a broad spectrum serine protease inhibitor that reduces eosinophil infiltration, mast cell activation and airway responsiveness in a murine model of asthma. Learn MoreStarting at: $45.00
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KU 60019
KU 60019 is a potent ATM kinase inhibitor with an IC50 value of 6.3 nM. Learn MoreStarting at: $189.00
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BC 11 hydrobromide
BC 11 hydrobromide is a selective urokinase (uPA) inhibitor (IC50 = 8.2 μM), which exhibits no activity at 8 other related enzymes, and inhibits clot lysis with no effect on clot formation. Learn MoreStarting at: $105.00
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4-Chlorophenylguanidine hydrochloride
4-Chlorophenylguanidine hydrochloride is a potent and specific inhibitor of urokinase. Learn MoreStarting at: $120.00
