Adrenergic Receptors
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A 80426 mesylate
A 80426 mesylate is a high affinity α2-adrenoceptor antagonist and selective 5-HT uptake inhibitor (Ki values are 2.01 and 3.77 nM respectively), which displays low affinity at a variety of structurally homologous GPCRs. Learn MoreStarting at: $115.00
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RS 79948 hydrochloride
RS 79948 hydrochloride is a α2-adrenoreceptor antagonist (Kd values are; 0.18, 0.19 and 0.42 nM for α2B α2C and α2A, respectively in rat). Learn MoreStarting at: $95.00
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RWJ 52353
RWJ 52353 is an agonist of the α2D adrenergic receptor (Ki values are 1.5, 254, 443 and 621 nM for α2D, α2A, α1 and α2B adrenergic receptors respectively). Learn MoreStarting at: $140.00
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Agmatine sulfate
Agmatine sulfate is a arginine metabolite that is synthesized within bovine brain and exhibits clonidine-displacing substance (CDS) activity. Learn MoreStarting at: $55.00
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Guanfacine hydrochloride
Guanfacine hydrochloride is a selective α2A-adrenoceptor agonist (Kd = 31 nM) which displays 60-fold selectivity over α2B-adrenoceptors. Learn MoreStarting at: $59.00
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Xamoterol hemifumarate
Xamoterol hemifumarate is a β1-adrenoceptor-selective partial agonist. Learn MoreStarting at: $109.00
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Betaxolol hydrochloride
Betaxolol hydrochloride is a selective β1-adrenoceptor antagonist. Learn MoreStarting at: $109.00
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Metoprolol tartrate
Metoprolol tartrate is a selective 1-adrenoceptor antagonist that inhibits spontaneous endothelin-1 production in vitro and displays antihypertensive and antianginal activity in vivo. Learn MoreStarting at: $55.00
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CGP 20712 dihydrochloride
CGP 20712 dihydrochloride is a highly selective and potent β1-adrenoceptor antagonist (IC50 = 0.7 nM), which displays 10,000-fold selectivity over β2-adrenoceptors. Learn MoreStarting at: $105.00
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Formoterol hemifumarate
Formoterol hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist which displays 330-fold selectivity for β2 over β1 receptors (pKd values are 8.12 and 5.58 respectively). Learn MoreStarting at: $70.00
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Zinterol hydrochloride
Zinterol hydrochloride is a potent and selective β2-adrenoceptor agonist (pKB values are 8.3 and < 5.7 for β 2 and β1 receptors respectively, as measured in human artery). Learn MoreStarting at: $119.00
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CGP 12177 hydrochloride
CGP 12177 hydrochloride is a partial agonist at β3-adrenoceptors. β1- and β2-adrenoceptor antagonist. Learn MoreStarting at: $55.00
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L-755,507
L-BMAA hydrochloride is a neurotoxic glutamate agonist originally isolated from Cycas circinalis. Learn MoreStarting at: $115.00
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(S)-(-)-Pindolol
(S)-(-)-Pindolol is a 5-HT1A/1Breceptor antagonist, with roughly equal affinity for each subtype. Learn MoreStarting at: $135.00
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L-748,337
L-748,337 is a competitive β3-adrenoceptor antagonist that displays selectivity over β1 and β2 receptors (Ki values are 4.0, 204 and 390 nM for β3-, β2- and β1-adrenoceptors respectively). Learn MoreStarting at: $119.00
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ZD 2079
β3-adrenoceptor agonist. Relaxes rat mesenteric artery and isolated aorta in vitro. Inhibits ob gene expression and circulating leptin levels in lean mice in vivo. Learn MoreStarting at: $95.00
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CL 316243 disodium salt
CL 316243 disodium salt is a potent and highly selective β3-adrenoceptor agonist (EC50 = 3 nM); > 10000-fold selective over β1 and β2 receptors. Learn MoreStarting at: $135.00
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ICI 215,001 hydrochloride
ICI 215,001 hydrochloride is the active metabolite of ZD 7114. Learn MoreStarting at: $105.00
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ZD 7114 hydrochloride
ZD 7114 hydrochloride is a β3-adrenoceptor agonist. Learn MoreStarting at: $100.00
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SR 58611A hydrochloride
Selective β3-adrenergic receptor agonist which displays both anxiolytic and antidepressant effects in rodent models. Learn MoreStarting at: $105.00