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5-HT Receptors
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4F 4PP oxalate
4F 4PP oxalate is a selective 5-HT2A antagonist with almost as high affinity (Ki = 5.3 nM) as ketanserin but with a much lower affinity for 5-HT2C sites (Ki = 620 nM). Learn MoreStarting at: $98.00
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S 14506 hydrochloride
S 14506 hydrochloride is a highly potent selective 5-HT1A receptor full agonist (pKi values are 9.0, 6.6, 7.5, 6.6 and < 6.0 for 5-HT1A, 5-HT1B, 5-HT1C, 5-HT2 and 5-HT3 receptors respectively). Learn MoreStarting at: $135.00
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Sarpogrelate hydrochloride
Sarpogrelate hydrochloride is a selective 5-HT2A receptor antagonist (pKi values are 8.52, 7.43 and 6.57 for 5-HT2A, 5-HT2C and 5-HT2B receptors respectively), which displays selectivity over 5-HT1, 5-HT3, 5-HT4 H1, H2, M3, α1-adrenergic, α2-adrenergic and β-adrenergic receptors. Learn MoreStarting at: $100.00
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DV 7028 hydrochloride
DV 7028 hydrochloride is a selective 5-HT2A receptor antagonist (Ki = 22 nM for at 5-HT2 receptors). Learn MoreStarting at: $105.00
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Fananserin
Fananserin is a 5-HT2A receptor antagonist that also displays high affinity at D4 receptors (Ki values are 0.26, 2.93, 25, 38, 70 and 726 nM for 5-HT2A, D4, H1, α1, 5-HT1A and D2 receptors respectively). Learn MoreStarting at: $95.00
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MDL 73005EF hydrochloride
MDL 73005EF hydrochloride is a potent and selective 5-HT1A receptor antagonist, which has partial agonist properties. Learn MoreStarting at: $90.00
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MDL 72832 hydrochloride
MDL 72832 hydrochloride is a potent ligand at 5-HT1A receptors, with mixed agonist and antagonist properties. Learn MoreStarting at: $90.00
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Altanserin hydrochloride
Altanserin hydrochloride is a potent and selective 5-HT2A receptor antagonist (Ki values are 0.13, 4.55, 40, 62 and 1570 nM at 5-HT2A, α1, 5-HT2C, D2 and 5-HT1A respectively). Learn MoreStarting at: $95.00
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MDL 11,939
MDL 11,939 is an Orally active 5-HT2A receptor antagonist, which displays selectivity for 5-HT2A receptors over 5-HT2C receptors (Ki values are 0.54, 2.5, 81.6 and ~10,000 nM at rabbit 5-HT2A, human 5-HT2A, rabbit 5-HT2C and human 5-HT2C receptors respectively). Learn MoreStarting at: $105.00
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Buspirone hydrochloride
Buspirone hydrochloride is a classic 5-HT1A partial agonist with relatively high affinity (Ki = 9.3 - 29.5 nM). Learn MoreStarting at: $49.00
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DOI hydrochloride
Brain penetrant, mixed 5-HT2A/5-HT2C receptor agonist (Ki values are 0.7, 2.4 and 20 nM for 5-HT2A, 5-HT2C and 5-HT2B receptors respectively), which reduces rapid eye movement (REM) and slow wave sleep and increases waking in the rat. Learn MoreStarting at: $90.00
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TCB-2
TCB-2 is a high affinity 5-HT2A receptor agonist that potently stimulates IP3 accumulation in NIH3T3 cells stably expressing rat 5-HT2A receptors with an EC50 value of 36 nM. Learn MoreStarting at: $139.00
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Xaliproden hydrochloride
Xaliproden hydrochloride is an orally active, full agonist at 5-HT1A receptors that is > 300-fold selective over other 5-HT receptor subtypes with an IC50 value of > 650 nM. Learn MoreStarting at: $105.00
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BP 554 maleate
BP 554 maleate is a selective 5-HT1A agonist. Learn MoreStarting at: $95.00
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Nefazodone hydrochloride
Nefazodone hydrochloride is a serotonin 5-HT2A receptor antagonist (Ki = 5.8 nM) and inhibitor of serotonin and noradrenalin uptake (IC50 values are 290 and 300 nM respectively). Learn MoreStarting at: $89.00
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(R)-(+)-8-Hydroxy-DPAT hydrobromide
(R)-(+)-8-Hydroxy-DPAT hydrobromide is a full 5-HT1A serotonin receptor agonist that reduces hippocampal 5-HT levels following systemic administration in rats in vivo. It is more active enantiomer of 8-Hydroxy-DPAT hydrobromide. Learn MoreStarting at: $109.00
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8-Hydroxy-DPAT hydrobromide
8-Hydroxy-DPAT hydrobromide is a standard selective 5-HT1A agonist that reduces hippocampal 5-HT levels following systemic administration in rats in vivo. Learn MoreStarting at: $59.00
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Spiperone hydrochloride
Spiperone hydrochloride is a 5-HT2A serotonin and selective D2-like dopamine receptor antagonist. Learn MoreStarting at: $99.00
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Mesulergine hydrochloride
Mesulergine hydrochloride is a 5-HT2A and 2C receptor antagonist and D2-like dopamine receptor partial agonist with antiprolactin and antiparkinsonian effects in vivo. Learn MoreStarting at: $129.00
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WAY 100635 maleate
WAY 100635 maleate is a potent, silent antagonist of 5-HT1A receptors with 100-fold selectivity for 5-HT1A over other 5-HT subtypes. It also has agonist activity at dopamine D4 receptors. Learn MoreStarting at: $119.00
