Transporters
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Org 25543 hydrochloride
Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2), which displays no activity at GlyT1 or 56 other common biological targets (≥ 100 μM), in a glycine uptake assay in CHO cells. Learn MoreStarting at: $139.00
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NFPS
NFPS is a selective, non-transportable inhibitor of GlyT1 which displays no activity on GlyT2 or the transport of proline, GABA or glutamate (IC50 values are 2.8, 9.8 and 56000 nM for hGlyT1, rGlyT1 and rGlyT2 respectively). Learn MoreStarting at: $139.00
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Sarcosine
Sarcosine is an endogenous inhibitor of GlyT1 that displays antipsychotic activity. Learn MoreStarting at: $55.00
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Dilazep dihydrochloride
Dilazep dihydrochloride is a coronary and cerebral vasodilator, suppresses the effects of ischemia. Learn MoreStarting at: $90.00
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N2-Methyl-L-arginine
N2-Methyl-L-arginine is a selective L-arginine uptake inhibitor (Ki = 500 μM) which inhibits uptake of arginine by the lysosomal system c in human fibroblast in vitro. Learn MoreStarting at: $119.00
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VU 0240551
VU 0240551 is an inhibitor of the neuronal K-Cl cotransporter, KCC2 that also inhibits hERG and L-type Ca2+ channels. Learn MoreStarting at: $115.00
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Decynium 22
Decynium 22 is an inhibitor of the plasma membrane monoamine transporter (PMAT) (Ki = 0.10 μM). Learn MoreStarting at: $49.00