Melatonin Receptors
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N-Acetyltryptamine
N-Acetyltryptamine is a partial agonist for melatonin receptors in the retina that also been used for determination of serotonin N-acetyl transferase. Learn MoreStarting at: $85.00
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Melatonin
Melatonin is an endogenous hormone that acts as an agonist at melatonin receptors MT1 and MT2. Learn MoreStarting at: $55.00
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6-Chloromelatonin
6-Chloromelatonin is a potent melatonin agonist with pKi values of 9.10 and 9.77 for human recombinant MT1 and MT2 receptors respectively. Learn MoreStarting at: $59.00
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DH 97
DH 97 is a relatively potent MT2 melatonin receptor antagonist (pKi value = 8.03), displaying 89- and 229-fold selectivity over MT1 and GPR50 (melatonin-related orphan receptor) respectively. Learn MoreStarting at: $98.00
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GR 135531
GR 135531 binds with high affinity to MT3 melatonin sites in hamster brain, and low affinity (and no efficacy) at MT1 and MT2 melatonin receptors and thus can be used to discriminate between the melatonin receptor subtypes. Learn MoreStarting at: $98.00
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2-Phenylmelatonin
2-Phenylmelatonin is a highly potent melatonin agonist which displays higher affinity and greater potency than melatonin itself. Learn MoreStarting at: $90.00
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4-P-PDOT
4-P-PDOT is a melatonin receptor antagonist, >300-fold selective for the MT2 (vs MT1) subtype. Learn MoreStarting at: $95.00
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8-M-PDOT
8-M-PDOT is a melatonin receptor agonist, 20-fold selective for the MT2 (vs MT1) subtype. Learn MoreStarting at: $95.00
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Luzindole
Luzindole is a melatonin antagonist. Learn MoreStarting at: $95.00
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2-Iodomelatonin
2-Iodomelatonin is a potent melatonin agonist with pKi values of 10.55 and 9.87 at human recombinant MT1 and MT2 receptors respectively. Learn MoreStarting at: $55.00