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Peptide Receptors
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CGP 71683 hydrochloride
Extremely selective, non-peptide NPY Y5 receptor antagonist. Displays > 1000-fold selectivity over Y1, Y2 and Y4 receptors; IC50 values are 1.4, 2765, 7187 and 5637 nM at cloned rat Y5, Y1, Y2 and Y4 receptors respectively. Learn MoreStarting at: $139.00
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BIBO 3304 trifluoroacetate
BIBO 3304 trifluoroacetate is a high affinity NPY Y1 receptor antagonist (IC50 values are 0.38 and 0.72 nM at human and rat receptors respectively) that displays > 2600-fold selectivity over Y2, Y4 and Y5 receptors. Learn MoreStarting at: $215.00
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BMS 193885
BMS 193885 is a potent, competitive neuropeptide (NPY) Y1 antagonist (Ki = 3.3 nM, IC50 = 5.9 nM) that displays > 47, > 100, > 160, > 160 and > 160-fold selectivity over σ1, α1, Y2, Y4 and Y5 receptors respectively. Learn MoreStarting at: $168.00
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PD 160170
PD 160170 is a potent, selective non-peptidic neuropeptide Y1 receptor antagonist (Ki = 48 nM); selective over Y2 and Y5 receptors (Ki > 10 μM). Learn MoreStarting at: $110.00
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CYM 9484
CYM 9484 is a potent neuropeptide Y (NPY) Y2 receptor antagonist (IC50 = 19 nM). Learn MoreStarting at: $140.00
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S 25585
S 25585 is a potent neuropeptide Y (NPY) Y5 receptor antagonist (IC50 values are 5.4, > 1000, > 10 000 and > 10 000 nM at Y5, Y1, Y2 and Y4 receptors respectively) that displays no affinity for a wide range of other receptors. Learn MoreStarting at: $139.00
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LU AA33810
LU AA33810 is a potent neuropeptide Y (NPY) Y5 receptor antagonist (Ki = 1.5 nM in vitro) which displays ≥ 3300-fold affinity for Y5 over Y1, Y2 and Y4 receptors. Learn MoreStarting at: $109.00
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NPY 5RA972
NPY 5RA972 is a potent and selective neuropeptide Y Y5 receptor antagonist (IC50 values are 3.1, >10000, >10000 and >10000 nM for Y5, Y1, Y2 and Y4 receptors respectively). Does not block NPY-induced feeding in vivo. Orally active and brain penetrant. Learn MoreStarting at: $135.00
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SF 11
SF 11 is a NPY Y2 antagonist (IC50 = 199 nM), which displays no affinity for Y1 receptor at concentrations up to 35 μM. Causes significant lethality in mice. Brain penetrant. Learn MoreStarting at: $139.00
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NTNCB hydrochloride
NTNCB hydrochloride is a selective, non-peptide competitive NPY Y5 antagonist. Ki values are 8.0 and 16032 nM at human recombinant Y5 and Y1 receptors respectively. Learn MoreStarting at: $149.00
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BIBP 3226 trifluoroacetate
3F8 is a potent and selective GSK-3β inhibitor (IC50 values are 34 and 304 nM in the presence of 10 and 100 μM ATP respectively). Learn MoreStarting at: $90.00
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L-152804
L-152804 is a potent, selective non-peptide neuropeptide Y Y5 receptor antagonist with > 300-fold selectivity over hY1, hY2, and hY4 receptors. Learn MoreStarting at: $145.00
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SR 142948
SR 142948 is a potent non-peptide neurotensin (NT) receptor antagonist that binds with high affinity (IC50 = 0.32 - 3.96 nM; Ki < 10 nM). Learn MoreStarting at: $85.00
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RF 9
RF 9 is a selective NPFF receptor antagonist that blocks NPFF-induced hypothermia and increases in atrial blood pressure and heart rate, and prevents opioid-induced tolerance associated with hyperalgesia in vivo. Learn MoreStarting at: $85.00
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BMS 470539 dihydrochloride
BMS 470539 dihydrochlorideis a potent, selective melanocortin MC1 receptor agonist (IC50 = 120 nM), which exhibits anti-inflammatory properties following ischemia-reperfusion in the vasculature. Learn MoreStarting at: $169.00
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TC-MCH 7c
TC-MCH 7c is a potent, selective melanin-concentrating hormone receptor 1 (MCH1R) antagonist. Learn MoreStarting at: $195.00
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GW 803430
GW 803430 is an orally active melanin-concentrating hormone receptor 1 (MCH1) antagonist (IC50 = 9.3 nM) with antiobesity and antidepressant-like effects in rats and mice.. Learn MoreStarting at: $150.00
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ATC 0175 hydrochloride
ATC 0175 hydrochloride is a potent, selective and orally active melanin-concentrating hormone receptor 1 (MCH1) antagonist (IC50 values are 13.5 and > 10000 nM for MCH1 and MCH2 receptors respectively). Learn MoreStarting at: $149.00
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ATC 0065
ATC 0065 is an orally active, potent and selective melanin-concentrating hormone receptor 1 (MCH1) antagonist (IC50 = 15.7 nM) that displays > 96-fold selectivity over MCH2. Learn MoreStarting at: $149.00
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SNAP 94847 hydrochloride
SNAP 94847 hydrochloride is a potent melanin-concentrating hormone receptor 1 (MCH1) antagonist (Ki = 2.2 nM, KD = 530 pM) that displays > 80-fold and > 500-fold selectivity over α1A and D2 receptors respectively. Learn MoreStarting at: $149.00
