ETA Receptors

FR 139317

FR 139317 is a highly potent and selective ETA endothelin receptor antagonist (Ki values are 1 nM and 7.3 μM at ETA and ETB subtypes respectively). Learn More

Starting at: $155.00

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BMS 182874 hydrochloride

BMS 182874 hydrochloride is a potent, selective and competitive non-peptide endothelin ETA receptor antagonist (Ki = 48 nM) which displays > 1000-fold selectivity over ETB receptors. Inhibits ET-1-induced pressor response following oral or intravenous administration in vivo and inhibits ET-1-induced longitudinal muscle contraction in the mouse colon in vitro. Learn More

Starting at: $140.00

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CI 1020

Flunitrazepam is a ligand at the GABAA receptor benzodiazepine modulatory site which exhibits hypnotic effects and also displays anxiolytic and sedative properties. Learn More

Starting at: $65.00

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