CRF1 Receptors

CP 376395 hydrochloride

CP 376395 hydrochloride is a potent and selective CRF1 receptor antagonist (Ki values are 12 and >10000 nM for CRF1 and CRF2 receptors respectively). Learn More

Starting at: $135.00

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NBI 27914 hydrochloride

NBI 27914 hydrochloride is a selective, non-peptide corticotropin-releasing factor1 (CRF1) receptor antagonist (Ki = 1.7 nM) which blocks behavioral seizures in vivo. Learn More

Starting at: $110.00

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SN 003

SN 003 is a reversible corticotropin releasing factor receptor 1 (CRF1) antagonist (Ki values are 3.4 and 7.9 nM at rat and human CRF1 respectively) that displays >1000-fold selectivity over CRF2 receptors. Learn More

Starting at: $140.00

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Antalarmin hydrochloride

Antalarmin hydrochloride is a non-peptide corticotropin-releasing hormone receptor 1 (CRF1) antagonist (Ki = 1 nM), which suppresses CRF-induced ACTH secretion and blocks CRF- and novelty-induced anxiety-like behavior in animal models of anxiety. Learn More

Starting at: $140.00

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NBI 35965 hydrochloride

NBI 35965 hydrochloride is a potent and selective corticotropin-releasing factor receptor 1 (CRF1) antagonist that inhibits cAMP accumulation and adrenocorticotropic hormone (ACTH) production in vitro and attenuates CRF and ACTH production in vivo. Learn More

Starting at: $158.00

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