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Ion Channels
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Eliprodil
Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site. Learn MoreStarting at: $90.00
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5,7-Dichlorokynurenic acid sodium salt
Sodium salt of 5,7-Dichlorokynurenic acid, a potent antagonist at the glycine site of the NMDA receptor (Ki = 79 nM vs. [3H]-glycine). Learn MoreStarting at: $65.00
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CGS 19755
CGS 19755 is a potent, competitive NMDA receptor antagonist. Learn MoreStarting at: $129.00
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L-Cysteinesulfinic acid
L-Cysteinesulfinic acid is a agonist at mGlu1a and mGlu5a subtypes expressed in clonal RGT cell lines. Also agonist at NMDA and PLD-coupled mGlu receptors. Learn MoreStarting at: $70.00
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Remacemide hydrochloride
Remacemide hydrochloride is a non-competitive NMDA receptor antagonist which blocks ion channel and allosteric modulatory site (IC50 = 8 - 68 mM). Learn MoreStarting at: $115.00
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(S)-(-)-HA-966
(S)-(-)-HA-966 is a possesses potent sedative and ataxic action, probably through disruption of striatal dopaminergic mechanisms. Learn MoreStarting at: $95.00
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HU 211
HU 211 is a NMDA antagonist (IC50 = 11 μM for inhibition of [3H]MK-801 binding to rat forebrain membranes), which exhibits beneficial effects in experimental models of multiple sclerosis, bacterial meningitis, septic shock, epilepsy, and traumatic and ischemic brain injury. Brain penetrant. Learn MoreStarting at: $270.00
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PPPA
PPPA is a competitive NMDA receptor antagonist that displays moderate selectivity for NR2A-containing receptors (Ki values are 0.13, 0.47, 1.10 and 3.86 μM for NR2A, NR2B, NR2C and NR2D subunits respectively). Learn MoreStarting at: $130.00
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PMPA (NMDA antagonist)
PMPA (NMDA antagonist) is a competitive NMDA receptor antagonist, which displays Ki values of 0.84, 2.74, 3.53 and 4.16 μM at NR2A, NR2B, NR2C and NR2D subunit-containing receptors respectively. Learn MoreStarting at: $125.00
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D-CPP-ene
D-CPP-ene is a potent and competitive NMDA antagonist (Ki = 40 nM). Learn MoreStarting at: $270.00
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DL-AP5 Sodium salt
DL-AP5 Sodium salt is a sodium salt of DL-AP5. Potent NMDA antagonist. Learn MoreStarting at: $69.00
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5,7-Dichlorokynurenic acid
5,7-Dichlorokynurenic acid is a potent antagonist at the glycine site of the NMDA receptor (Ki = 79 nM vs. [3H]-glycine). Learn MoreStarting at: $65.00
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SDZ 220-040
SDZ 220-040 is a potent competitive antagonist at the NMDA receptor (pKi = 8.5). Learn MoreStarting at: $140.00
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D-Aspartic acid
Endogenous NMDA receptor agonist with similar activity to the L-isomer (L-aspartic acid). Learn MoreStarting at: $80.00
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AR-R 17779 hydrochloride
AR-R 17779 hydrochloride is a selective agonist of α7 nAChRs (Ki values are 190 and 16000 nM for rat α7 and α4β2 receptors respectively). Learn MoreStarting at: $140.00
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Co 101244 hydrochloride
Co 101244 hydrochloride is a novel, potent and selective antagonist of NR2B-containing NMDA receptors (IC50 values are 0.043, > 100 and > 100 μM for NR1A/2B, NR1A/2A and NR1A/2C subunit combinations respectively). Learn MoreStarting at: $119.00
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Ro 04-5595 hydrochloride
Ro 04-5595 hydrochloride is a selective antagonist for NR2B-containing NMDA receptors (Ki = 31 nM). Learn MoreStarting at: $129.00
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Ro 8-4304 hydrochloride
Ro 8-4304 hydrochloride is a NMDA receptor antagonist (IC50 = 0.4 μM) that displays > 100 fold selectivity for NR2B-containing receptors over NR2A-containing receptors, which exhibits an activity-dependent mechanism of NMDA antagonism and is competitive with respect to spermine. Learn MoreStarting at: $109.00
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CGP 78608 hydrochloride
CGP 78608 hydrochloride is a potent and selective NMDA antagonist that acts through the glycine site (IC50 = 5 nM). Displays > 500-fold selectivity over kainate and AMPA receptors (IC50 values are 2.7 and 3 μM respectively). Learn MoreStarting at: $140.00
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ACBC
ACBC is a NMDA receptor partial agonist, acting at the glycine site of NR1. Learn MoreStarting at: $80.00
