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Glutamate (Ionotropic) Receptors
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Pentamidine isethionate
Antimicrobial. Neuroprotective; inhibits constitutive nitric oxide synthase in the brain and acts as a NMDA glutamate receptor antagonist. Learn MoreStarting at: $80.00
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CGP 78608 hydrochloride
CGP 78608 hydrochloride is a potent and selective NMDA antagonist that acts through the glycine site (IC50 = 5 nM). Displays > 500-fold selectivity over kainate and AMPA receptors (IC50 values are 2.7 and 3 μM respectively). Learn MoreStarting at: $140.00
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DQP 1105
DQP 1105 is a noncompetitive NMDA receptor antagonist; displays over 50-fold selectivity for GluN2D- and GluN2C-containing receptors over GluN2B-, GluK2-, GluA1- and GluN2A-containing receptors (IC50 values are 2.7, 8.5, 121, 153, 198 and 206 μM respectively). Learn MoreStarting at: $119.00
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ACBC
ACBC is a NMDA receptor partial agonist, acting at the glycine site of NR1. Learn MoreStarting at: $80.00
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Ifenprodil hemitartrate
Ifenprodil hemitartrate is a NMDA receptor antagonist, acting at the polyamine site. Learn MoreStarting at: $65.00
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Synthalin sulfate
Synthalin sulfate is an effective non-competitive NMDA receptor antagonist in vivo and in vitro. Learn MoreStarting at: $85.00
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TCS 46b
Orally active, subtype-selective NR1A/NR2B NMDA receptor antagonist (IC50 values are 5.3, 35000 and > 100000 nM for NR1A/2B, NR1A/2A and NR1A/2C receptor subtypes respectively), whih potentiates the effect of L-DOPA in 6-OHDA-lesioned rats following oral administration. Learn MoreStarting at: $109.00
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Spermine tetrahydrochloride
Spermine tetrahydrochloride is a polyamine which produces a variety of modulatory effects on the NMDA receptor channel, acting through a specific site on the complex which can cause both agonist and antagonist effects. Learn MoreStarting at: $59.00
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D-Serine
D-Serine is a glycine agonist at the NMDA receptor. L-Serine also available. Learn MoreStarting at: $79.00
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Ro 8-4304 hydrochloride
Ro 8-4304 hydrochloride is a NMDA receptor antagonist (IC50 = 0.4 μM) that displays > 100 fold selectivity for NR2B-containing receptors over NR2A-containing receptors, which exhibits an activity-dependent mechanism of NMDA antagonism and is competitive with respect to spermine. Learn MoreStarting at: $109.00
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Ro 04-5595 hydrochloride
Ro 04-5595 hydrochloride is a selective antagonist for NR2B-containing NMDA receptors (Ki = 31 nM). Learn MoreStarting at: $129.00
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(2R,3S)-Chlorpheg
(2R,3S)-Chlorpheg is a weakly active NMDA receptor antagonist. Learn MoreStarting at: $185.00
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L-701,324
L-701,324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor. Learn MoreStarting at: $95.00
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Arcaine sulfate
Arcaine sulfate is a NO synthase inhibitor, acting as a competitive inhibitor at the polyamine site. Learn MoreStarting at: $80.00
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L-701,252
L-701,252 is an antagonist at the glycine-NMDA site (IC50 = 420 nM). Learn MoreStarting at: $95.00
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Gavestinel
Gavestinel is a highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM), which displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites. Orally bioavailable and active in vivo. Learn MoreStarting at: $100.00
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SDZ 220-040
SDZ 220-040 is a potent competitive antagonist at the NMDA receptor (pKi = 8.5). Learn MoreStarting at: $140.00
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D-Aspartic acid
Endogenous NMDA receptor agonist with similar activity to the L-isomer (L-aspartic acid). Learn MoreStarting at: $80.00
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Co 101244 hydrochloride
Co 101244 hydrochloride is a novel, potent and selective antagonist of NR2B-containing NMDA receptors (IC50 values are 0.043, > 100 and > 100 μM for NR1A/2B, NR1A/2A and NR1A/2C subunit combinations respectively). Learn MoreStarting at: $119.00
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Spermidine trihydrochloride
Spermidine trihydrochloride binds to the polyamine modulatory site of the NMDA receptor and has been described as an agonist based on its ability to enhance the binding of [3H]-MK801. Learn MoreStarting at: $65.00
