Proteases
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ZJ 43
ZJ 43 is a potent inhibitor of glutamate carboxypeptidase II and III (GCP II and III/NAAG peptidase/NAALADase) that inhibits the hydrolysis of NAAG (IC50 = 2.4 nM). Learn MoreStarting at: $89.00
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PMPA (NAALADase inhibitor)
PMPA (NAALADase inhibitor) is a highly potent and selective inhibitor of glutamate carboxypeptidase 2 (GCP II/N-acetylated α-linked dipeptidase/NAALADase) with a Ki value of 275 pM. Learn MoreStarting at: $90.00
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Captopril
Captopril is a angiotensin-converting enzyme (ACE) inhibitor that also displays reversible, competitive inhibition of leukotriene A4 (LTA4) hydrolase. Learn MoreStarting at: $38.00
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Moexipril hydrochloride
Moexipril hydrochloride is an angiotensin-converting enzyme (ACE) inhibitor that decreases mean blood pressure in the spontaneous hypertensive rat (SHR) and also blocks degradation of bradykinin into inactive metabolites. Learn MoreStarting at: $109.00
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Fumagillin
Fumagillin is an antibiotic and antiangiogenic agent, which covalently binds and inhibits methionine aminopeptidase-2. Learn MoreStarting at: $119.00
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SID 26681509
SID 26681509 is a potent and reversible human cathepsin L inhibitor with an IC50 value of 56 nM. Learn MoreStarting at: $149.00
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L 006235
L 006235 is a potent, reversible cathepsin K inhibitor (IC50 = 0.25 nM) that displays > 4000-fold selectivity over cathepsins B, L and S. Learn MoreStarting at: $159.00
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N-Acetyl-L-leucyl-L-leucyl-L-methional
N-Acetyl-L-leucyl-L-leucyl-L-methional is a very potent inhibitor of cathepsin L (Ki = 0.6 nM) and the strongest inhibitor of cathepsin B (Ki = 100 nM) amongst the peptide aldehydes. Learn MoreStarting at: $90.00
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PD 150606
PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively). Learn MoreStarting at: $100.00