Opioid Receptors
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Naltrindole hydrochloride
Naltrindole hydrochloride is a highly selective non-peptide δ opioid antagonist, showing 223- and 346-fold greater activity at δ than at μ and κ opioid receptors. Learn MoreStarting at: $95.00
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FIT
FIT is a selective and irreversible δ-opioid agonist that acts by alkylating the receptor. Learn MoreStarting at: $139.00
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SDM25N hydrochloride
SDM25N hydrochloride is a potent and highly selective non-peptide δ receptor antagonist (Ki values are 4.7, 3800 and 7900 nM for δ, κ and μ receptors respectively). Learn MoreStarting at: $125.00
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AR-M 1000390 hydrochloride
AR-M 1000390 hydrochloride is a non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80. Learn MoreStarting at: $119.00
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SNC 162
SNC 162 is a potent and selective non-peptide δ-opioid receptor agonist (Ki = 0.63 nM) which displays > 8000-fold selectivity over μ-opioid receptors and is centrally active following systemic administration in vivo. Learn MoreStarting at: $160.00
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SNC 80
SNC 80 is a highly selective and potent non-peptide δ-opioid agonist, 2000-fold selective over μ-opioid receptors. Learn MoreStarting at: $140.00
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BW 373U86
BW 373U86 is a potent, selective non-peptide δ-opioid receptor agonist. Learn MoreStarting at: $200.00
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SB 205607 dihydrobromide
SB 205607 dihydrobromide is the first described non-peptide δ1 opioid receptor agonist with very high affinity and selectivity for the δ1 subtype (Ki values are 1.12, 2320 and 1790 nM at δ1, μ and κ receptors respectively). Learn MoreStarting at: $175.00
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BNTX maleate
BNTX maleate is a standard selective δ1 opioid receptor antagonist, which inhibits neurogenic ion transport mediated by a putative novel opioid receptor in porcine ileal mucosa. Learn MoreStarting at: $115.00
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N-Benzylnaltrindole hydrochloride
N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist with a long duration of action in vivo. Learn MoreStarting at: $95.00
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Naltriben mesylate
Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively), which displays selectivity for the δ2 subtype in vivo. Learn MoreStarting at: $100.00
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GNTI dihydrochloride
GNTI dihydrochloride is a highly potent κ opioid receptor antagonist (Ki = 0.18 nM for human cloned κ receptors expressed in CHO cells), which displays 208- and 799-fold selectivity over μ and δ receptors respectively. Learn MoreStarting at: $139.00
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(±)-U-50488 hydrochloride
(±)-U-50488 hydrochloride is as elective κ-opioid agonist. Learn MoreStarting at: $99.00
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(+)-U-50488 hydrochloride
(+)-U-50488 hydrochloride is a less active enantiomer of (±)-U-50488. Learn MoreStarting at: $98.00
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(-)-U-50488 hydrochloride
(-)-U-50488 hydrochloride is a more active enantiomer of (±)-U-50488. Learn MoreStarting at: $99.00
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Salvinorin A
Salvinorin A displays high affinity at both native (Ki = 4.3 nM) and cloned (Ki = 16 nM) κ-opioid receptors. Learn MoreStarting at: $139.00
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N-MPPP Hydrochloride
N-MPPP Hydrochloride is a high affinity κ agonist with no measured binding at μ or δ sites. Learn MoreStarting at: $110.00
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DIPPA hydrochloride
DIPPA hydrochloride is an irreversible and selective antagonist at the κ receptor, with persistent effect in vivo. Learn MoreStarting at: $100.00
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GR 89696 fumarate
Highly potent and selective κ-opioid agonist (IC50 = 0.04 nM) that may be selective for the putative κ2 receptor. Learn MoreStarting at: $135.00
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ICI 204,448 hydrochloride
ICI 204,448 hydrochloride is a peripherally acting κ agonist. Learn MoreStarting at: $95.00