Opioid Receptors
-
ICI 199,441 hydrochloride
ICI 199,441 hydrochloride is a highly potent κ agonist, 146-fold more active than U-50488 in vitro. Learn MoreStarting at: $95.00
-
U-54494A hydrochloride
U-54494A hydrochloride is a κ-opioid agonist and anticonvulsant, which acts as an NMDA antagonist. Learn MoreStarting at: $105.00
-
nor-Binaltorphimine dihydrochloride
nor-Binaltorphimine dihydrochloride is a selective κ-opioid receptor antagonist. Learn MoreStarting at: $90.00
-
Fentanyl citrate
Fentanyl citrate is a potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively), which displays antinociceptive activity in vivo. Learn MoreStarting at: $55.00
-
Etonitazenyl isothiocyanate
Etonitazenyl isothiocyanate is an affinity label specific for μ opioid sites. Learn MoreStarting at: $125.00
-
Naloxonazine dihydrochloride
Naloxonazine dihydrochloride is a potent opioid antagonist, selective for μ1 receptors. Learn MoreStarting at: $79.00
-
β-Funaltrexamine hydrochloride
β-Funaltrexamine hydrochloride is a selective μ opioid receptor antagonist. Learn MoreStarting at: $149.00
-
Oxycodone hydrochloride
Oxycodone hydrochloride is a potent and selective μ-opioid receptor agonist (Ki values are 16 and >1000 nM for hMOR1 and hKOR1 respectively). Learn MoreStarting at: $65.00
-
Cyprodime hydrochloride
Cyprodime hydrochloride is a selective μ-opioid receptor antagonist (Ki values are 5.4, 244.6 and 2187 nM for μ-, δ- and κ-opioid receptors respectively). Learn MoreStarting at: $130.00
-
Clocinnamox mesylate
Clocinnamox mesylate is a systemically active, irreversible μ-opioid receptor antagonist (apparent Ki values are 0.7, 1.9 and 5.7 nM for mouse μ, δ and κ receptors respectively). Learn MoreStarting at: $95.00
-
Trap 101
Trap 101 is a potent and selective nociceptin/orphanin FQ (NOP) receptor antagonist. Learn MoreStarting at: $139.00
-
SB 612111 hydrochloride
SB 612111 hydrochloride is a selective NOP receptor antagonist (Ki values are 0.33, 57.6, 160.5 and 2109 nM for NOP, μ-, κ- and δ-receptors respectively), which antagonizes the pronociceptive action of nociceptin in an acute pain model. Learn MoreStarting at: $179.00
-
SCH 221510
SCH 221510 is a potent and selective nociceptin opioid receptor (NOP) agonist (EC50 values are 12, 693, 683 and 8071 nM, and Ki values are 0.3, 65, 131 and 2854 nM at NOP, μ-, κ- and δ-opioid receptors respectively). Learn MoreStarting at: $145.00
-
NNC 63-0532
NNC 63-0532 is a potent non-peptide agonist for the NOP receptor (EC50 = 305 nM, Ki = 7.3 nM); ~ 12-fold selective over other receptors. Learn MoreStarting at: $155.00
-
(±)-J 113397
(±)-J 113397 is a potent and selective NOP receptor antagonist (IC50 values are 2.3, 1400, 2200 and > 10000 nM for NOP, κ, μ and δ-opioid receptors respectively), which inhibits nociceptin/orphanin FQ-induced hyperalgesia in the mouse tail-flick test. Learn MoreStarting at: $189.00
-
Naloxone benzoylhydrazone
Naloxone benzoylhydrazone is a mixed opioid receptor agonist/antagonist. Learn MoreStarting at: $80.00
-
Diprenorphine
Diprenorphine is a non-selective opioid receptor antagonist (Ki values are 0.017, 0.072 and 0.23 nM for κ-, μ- and δ-opioid receptors). Learn MoreStarting at: $125.00
-
Naloxone hydrochloride
Naloxone hydrochloride is an opioid antagonist. Learn MoreStarting at: $79.00
-
Naltrexone hydrochloride
Doxepin hydrochloride is a highly potent H1 histamine receptor antagonist (Kd = 310 pM) and tricyclic antidepressant. Learn MoreStarting at: $50.00
-
Buprenorphine hydrochloride
Buprenorphine hydrochloride, an ORL1 receptor agonist, displays mixed antagonist/partial agonist activity at κ, δ and μ-opioid receptors. Learn MoreStarting at: $40.00