You have no items in your shopping cart.
Glutamate (Ionotropic) Receptors
-
5,7-Dichlorokynurenic acid sodium salt
Sodium salt of 5,7-Dichlorokynurenic acid, a potent antagonist at the glycine site of the NMDA receptor (Ki = 79 nM vs. [3H]-glycine). Learn MoreStarting at: $65.00
-
D-CPP-ene
D-CPP-ene is a potent and competitive NMDA antagonist (Ki = 40 nM). Learn MoreStarting at: $270.00
-
PMPA (NMDA antagonist)
PMPA (NMDA antagonist) is a competitive NMDA receptor antagonist, which displays Ki values of 0.84, 2.74, 3.53 and 4.16 μM at NR2A, NR2B, NR2C and NR2D subunit-containing receptors respectively. Learn MoreStarting at: $125.00
-
PPPA
PPPA is a competitive NMDA receptor antagonist that displays moderate selectivity for NR2A-containing receptors (Ki values are 0.13, 0.47, 1.10 and 3.86 μM for NR2A, NR2B, NR2C and NR2D subunits respectively). Learn MoreStarting at: $130.00
-
HU 211
HU 211 is a NMDA antagonist (IC50 = 11 μM for inhibition of [3H]MK-801 binding to rat forebrain membranes), which exhibits beneficial effects in experimental models of multiple sclerosis, bacterial meningitis, septic shock, epilepsy, and traumatic and ischemic brain injury. Brain penetrant. Learn MoreStarting at: $270.00
-
(S)-(-)-HA-966
(S)-(-)-HA-966 is a possesses potent sedative and ataxic action, probably through disruption of striatal dopaminergic mechanisms. Learn MoreStarting at: $95.00
-
Remacemide hydrochloride
Remacemide hydrochloride is a non-competitive NMDA receptor antagonist which blocks ion channel and allosteric modulatory site (IC50 = 8 - 68 mM). Learn MoreStarting at: $115.00
-
L-Cysteinesulfinic acid
L-Cysteinesulfinic acid is a agonist at mGlu1a and mGlu5a subtypes expressed in clonal RGT cell lines. Also agonist at NMDA and PLD-coupled mGlu receptors. Learn MoreStarting at: $70.00
-
CGS 19755
CGS 19755 is a potent, competitive NMDA receptor antagonist. Learn MoreStarting at: $129.00
-
(RS)-CPP
(RS)-CPP is a potent NMDA antagonist. Separate isomer (R)-CPP also available. Learn MoreStarting at: $129.00
-
(R)-CPP
(R)-CPP is a highly potent NMDA antagonist, which shows some selectivity for NR2A-containing receptors (Ki values are 0.041, 0.27, 0.63 and 1.99 μM for inhibition of NR2A-, NR2B-, NR2C- and NR2D-containing recombinant NMDA receptors respectively). Learn MoreStarting at: $245.00
-
CGP 37849
CGP 37849 is a potent, selective and competitive NMDA receptor antagonist (Ki = 35 nM). Learn MoreStarting at: $115.00
-
CGP 39551
CGP 39551 is a potent, selective and competitive NMDA antagonist (Ki = 310 nM for inhibition of [3H]-CPP binding in rat brain). Learn MoreStarting at: $115.00
-
SDZ 220-040
SDZ 220-040 is a potent competitive antagonist at the NMDA receptor (pKi = 8.5). Learn MoreStarting at: $140.00
-
Gavestinel
Gavestinel is a highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM), which displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites. Orally bioavailable and active in vivo. Learn MoreStarting at: $100.00
-
L-701,252
L-701,252 is an antagonist at the glycine-NMDA site (IC50 = 420 nM). Learn MoreStarting at: $95.00
-
Arcaine sulfate
Arcaine sulfate is a NO synthase inhibitor, acting as a competitive inhibitor at the polyamine site. Learn MoreStarting at: $80.00
-
L-701,324
L-701,324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor. Learn MoreStarting at: $95.00
-
(2R,3S)-Chlorpheg
(2R,3S)-Chlorpheg is a weakly active NMDA receptor antagonist. Learn MoreStarting at: $185.00
-
Pentamidine isethionate
Antimicrobial. Neuroprotective; inhibits constitutive nitric oxide synthase in the brain and acts as a NMDA glutamate receptor antagonist. Learn MoreStarting at: $80.00
