D3 Receptors
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SB 277011A dihydrochloride
SB 277011A dihydrochloride is a selective dopamine D3 receptor antagonist (pKi values are 8.0, 6.0, 5.0 and <5.2 for D3, D2, 5-HT1D and 5-HT1B respectively). Learn MoreStarting at: $115.00
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GSK 789472 hydrochloride
GSK 789472 hydrochloride is a selective dopamine D3 receptor antagonist and D2 partial agonist (pEC50 values are <5.5 and 8.3 respectively), which selective against the D4 receptor in both agonist and antagonist assays. Brain penetrant. Learn MoreStarting at: $95.00
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Nafadotride
Nafadotride is a highly potent, competitive, preferential dopamine D3 receptor antagonist. Ki values are 0.52, 5, and 269 nM for human cloned D3, D2 and D4 receptors respectively. Learn MoreStarting at: $135.00
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NGB 2904
NGB 2904 is a potent and selective dopamine D3 receptor antagonist (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4, D1 and D5 receptors respectively). Learn MoreStarting at: $135.00
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PNU 177864 hydrochloride
PNU 177864 hydrochloride is a highly selective dopamine D3 receptor antagonist which induces phospholipidosis and exhibits antischizophrenic activity in vivo. Learn MoreStarting at: $109.00
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7-Hydroxy-PIPAT maleate
8-Hydroxy-PIPAT oxalate is a high affinity 5-HT1A receptor agonist (Kd = 0.38 nM). Learn MoreStarting at: $120.00
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PG 01037 dihydrochloride
PG 01037 dihydrochloride is a Dopamine D3 receptor antagonist with 133-fold selectivity for D3 over D2 receptors in vitro (Ki values are 0.70, 93.3 and 375 nM for D3, D2 and D4 receptors respectively). Learn MoreStarting at: $139.00
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7-Hydroxy-DPAT hydrobromide
7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist. Learn MoreStarting at: $59.00
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U 99194 maleate
U 99194 maleateis a potent, selective D3 antagonist. Learn MoreStarting at: $109.00