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Cannabinoid Receptors
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Arvanil
Arvanil is a cannabinoid CB1 and vanilloid TRPV1 (VR1) agonist (Ki values are 0.5 and 0.3 μM respectively), which also inhibits the anandamide transporter (IC50 = 3.6 μM). Learn MoreStarting at: $50.00
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ACEA
ACEA is a potent and highly selective CB1 receptor agonist (Ki = 1.4 nM) which displays >1400-fold selectivity over CB2 receptors. Learn MoreStarting at: $55.00
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Noladin ether
Noladin ether is an endogenous agonist for the GPR55 and CB1 receptors (EC50 values are 10 and 37 nM respectively) that displays selectivity over CB2 receptors (Ki values are 21.2 nM and > 3mM at CB1 and CB2 respectively). Learn MoreStarting at: $98.00
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ACPA
ACPA is a potent and selective CB1 agonist (Ki = 2.2 nM) which displays 325-fold selectivity over CB2 receptors. Learn MoreStarting at: $69.00
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Oleamide
Oleamide endogenous sleep-inducing lipid, which acts as an agonist at the CB1 cannabinoid receptor (EC50 = 1.64 μM). Learn MoreStarting at: $59.00
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NIDA 41020
NIDA 41020 is a high affinity CB1 receptor antagonist (Ki = 4.1 nM), which exhibits significantly reduced lipophilicity compared to other CB1 antagonists. Learn MoreStarting at: $139.00
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TC-C 14G
TC-C 14G is a potent, high affinity CB1 receptor inverse agonist with high efficacy in a hypothermia assay (ID50 = 5 mg/kg) in vivo. Learn MoreStarting at: $140.00
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(±)-CP 47497
(±)-CP 47497 is a potent CB1 receptor agonist (Ki = 2.2 nM)that exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo. Learn MoreStarting at: $99.00
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PF 514273
PF 514273 is a potent and selective CB1 receptor antagonist that inhibits food intake in vivo following oral administration. Learn MoreStarting at: $139.00
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MJ 15
MJ 15 is a potent and selective CB1 receptor antagonist that inhibits food intake and increases in body weight in diet-induced obese rats and mice. Learn MoreStarting at: $139.00
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GGTI 297
GGTI 297 is a geranylgeranyltransferase I (GGTase-I) inhibitor (IC50 values are 135 and 418 nM for GGTase-I and FTase inhibition respectively), which inhibits RhoA prenylation leading to inactivation of RhoA/ROCK and a decrease in basal tone of the internal anal sphincter in vitro. Learn MoreStarting at: $149.00
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Tocrifluor T1117
Tocrifluor T1117 is a novel fluorescent form of AM 251, which conjugated with 5-carboxytetramethylrhodamine (5-TAMRA) that fluoresces at 543nm excitation (590nm emission), and displays GPR55 binding activity. Learn MoreStarting at: $200.00
