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Cannabinoid Receptors
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Palmitoylethanolamide
Palmitoylethanolamide, a selective GPR55 agonist, is a substrate for fatty acid amide hydrolase (FAAH) and PEA-preferring acid amidase (PAA) and exhibits antinociceptive and anticonvulsant in vivo. Learn MoreStarting at: $65.00
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CID 16020046
CID 16020046 is a selective GPR55 antagonist that inhibits LPI-induced Ca2+ signaling with an IC50 value of 0.21 μM in HEK-GPR55 cells. Learn MoreStarting at: $139.00
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Oleylethanolamide
Oleylethanolamide is a lipid mediator and analog of anandamide that is involved in peripheral regulation of feeding, which induces satiety through activation of PPARα and is also a ceramidase inhibitor. Learn MoreStarting at: $60.00
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GP 2a
GP 2a is a selective CB2 receptor agonist with Ki values of 7.6 and 900 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $169.00
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L-759,633
L-759,633 is a high affinity, selective CB2 receptor agonist (Ki values are 6.4 and 1043 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 8.1 nM). Learn MoreStarting at: $180.00
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CB 65
CB 65 is a high affinity and selective CB2 receptor agonist. Learn MoreStarting at: $139.00
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GP 1a
GP 1a is a highly selective CB2 receptor agonist that increases P-ERK1/2 expression in HL-60 cells in vitro with Ki values are 0.037 and 363 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $150.00
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AM 630
Immepip dihydrobromide is a potent histamine H3 receptor agonist which also binds to H4 receptors (Ki values are 0.4 and 9 nM at human recombinant H3 and H4 receptors respectively). Learn MoreStarting at: $135.00
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SER 601
SER 601 is a potent and selective CB2 receptor agonist (Ki values are 6.3 nM and 1.2 μM for CB2 and CB1 receptors respectively). Learn MoreStarting at: $109.00
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JWH 015
JWH 015 is a selective CB2 agonist (Ki values are 13.8 and 383 nM as measured at human cloned CB2 and CB1 receptors expressed in CHO cells). Learn MoreStarting at: $50.00
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L-759,656
Highly selective CB2 receptor agonist (Ki values are 11.8 and 4888 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 3.1 nM). Learn MoreStarting at: $180.00
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GW 405833
GW 405833 is a potent and selective CB2 receptor partial agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%) which binds with high affinity to both human and rat CB2 receptors and displays ~ 1200-fold selectivity over CB1 (Ki values are 3.92 and 4772 nM for human recombinant CB2 and CB1 receptors respectively). Learn MoreStarting at: $135.00
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HU 308
HU 308 is a potent and selective CB2 receptor agonist (Ki values are 22.7 nM and > 10 μM for CB2 and CB1 receptors respectively, EC50 = 5.57 nM) which displays antiallodynic activity in the rat hindpaw incision model of postoperative pain. Learn MoreStarting at: $179.00
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JTE 907
JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist, which binds with high affinity to rat, mouse and human CB2 receptors (Ki values are 0.38, 1.55 and 35.9 nM respectively). Learn MoreStarting at: $139.00
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AM 281
AM 281 is a potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively), which increases locomotor activity following systemic administration in vivo. Learn MoreStarting at: $140.00
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NADA
NADA is a potent endogenous cannabinoid and vanilloid receptor agonist, with no action at dopamine receptors. Selective for CB1 over CB2 receptors (Ki values are 0.25 and 12 μM respectively), and potent agonist at TRPV1 (VR1) receptors (EC50 ~ 50 nM). Learn MoreStarting at: $79.00
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LY 320135
LY 320135 is a potent CB1 receptor antagonist/inverse agonist (Ki = 141 nM) with greater than 70-fold selectivity over CB2 receptors (Ki > 10 μM). Learn MoreStarting at: $135.00
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(R)-(+)-Methanandamide
(R)-(+)-Methanandamide is a stable anandamide analog that is a selective agonist for the CB1 receptor (Ki values are 20 and 815 nM for CB1 and CB2 receptors respectively), which also displays agonist activity at vanilloid receptors. Learn MoreStarting at: $65.00
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DEA
DEA is a potent endocannabinoid and anandamide analog that activates CB1 receptors in microglia and binds to rat synaptosomal membranes (Ki = 34.4 nM). Learn MoreStarting at: $80.00
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Leelamine hydrochloride
Leelamine hydrochloride is a CB1 agonist which displaces binding of [3H]-SR141716A with an IC50 value of 2.86 μM. Learn MoreStarting at: $90.00
