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Cannabinoid Receptors
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GP 1a
GP 1a is a highly selective CB2 receptor agonist that increases P-ERK1/2 expression in HL-60 cells in vitro with Ki values are 0.037 and 363 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $150.00
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AM 630
Immepip dihydrobromide is a potent histamine H3 receptor agonist which also binds to H4 receptors (Ki values are 0.4 and 9 nM at human recombinant H3 and H4 receptors respectively). Learn MoreStarting at: $135.00
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JTE 907
JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist, which binds with high affinity to rat, mouse and human CB2 receptors (Ki values are 0.38, 1.55 and 35.9 nM respectively). Learn MoreStarting at: $139.00
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HU 308
HU 308 is a potent and selective CB2 receptor agonist (Ki values are 22.7 nM and > 10 μM for CB2 and CB1 receptors respectively, EC50 = 5.57 nM) which displays antiallodynic activity in the rat hindpaw incision model of postoperative pain. Learn MoreStarting at: $179.00
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GW 405833
GW 405833 is a potent and selective CB2 receptor partial agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%) which binds with high affinity to both human and rat CB2 receptors and displays ~ 1200-fold selectivity over CB1 (Ki values are 3.92 and 4772 nM for human recombinant CB2 and CB1 receptors respectively). Learn MoreStarting at: $135.00
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L-759,656
Highly selective CB2 receptor agonist (Ki values are 11.8 and 4888 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 3.1 nM). Learn MoreStarting at: $180.00
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L-759,633
L-759,633 is a high affinity, selective CB2 receptor agonist (Ki values are 6.4 and 1043 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 8.1 nM). Learn MoreStarting at: $180.00
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JWH 015
JWH 015 is a selective CB2 agonist (Ki values are 13.8 and 383 nM as measured at human cloned CB2 and CB1 receptors expressed in CHO cells). Learn MoreStarting at: $50.00
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SER 601
SER 601 is a potent and selective CB2 receptor agonist (Ki values are 6.3 nM and 1.2 μM for CB2 and CB1 receptors respectively). Learn MoreStarting at: $109.00
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CID 16020046
CID 16020046 is a selective GPR55 antagonist that inhibits LPI-induced Ca2+ signaling with an IC50 value of 0.21 μM in HEK-GPR55 cells. Learn MoreStarting at: $139.00
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Palmitoylethanolamide
Palmitoylethanolamide, a selective GPR55 agonist, is a substrate for fatty acid amide hydrolase (FAAH) and PEA-preferring acid amidase (PAA) and exhibits antinociceptive and anticonvulsant in vivo. Learn MoreStarting at: $65.00
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O-1602
O-1602 is an analog of cannabidiol that is a potent agonist at the GPR55 cannabinoid receptor (EC50 values are 13, > 30000 and > 30000 nM for GPR55, CB1 and CB2 receptors respectively). Learn MoreStarting at: $145.00
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Abn-CBD
Neurobehaviorally inactive cannabinoid that acts as a selective agonist for GPR55 (EC50 values are 2.5, >30 and >30 μM at GPR55, CB1 and CB2 receptors respectively). Learn MoreStarting at: $179.00
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Oleylethanolamide
Oleylethanolamide is a lipid mediator and analog of anandamide that is involved in peripheral regulation of feeding, which induces satiety through activation of PPARα and is also a ceramidase inhibitor. Learn MoreStarting at: $60.00
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Anandamide - d4
Anandamide - d4 is a deuterated anandamide that is used as an internal standard for the quantification of AEA by GC- or LC-mass spectrometry. Learn MoreStarting at: $149.00
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O-2545 hydrochloride
O-2545 hydrochloride is a high affinity, water-soluble CB1/CB2 receptor agonist. Learn MoreStarting at: $105.00
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CP 55940
CP 55940 is a cannabinoid agonist that displays high and roughly equal affinity for both central and peripheral cannabinoid receptors. Learn MoreStarting at: $189.00
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2-Arachidonylglycerol
2-Arachidonylglycerol is a endogenous cannabinoid ligand that acts as a potent agonist at GPR55 (EC50 values are 3, 519 and 618 nM at GPR55, CB1 and CB2 respectively; Ki values are 472 and 1400 nM at CB1 and CB2 respectively). Learn MoreStarting at: $132.00
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Cannabinol
Cannabinol, a CB2 and CB1 receptor agonist, inhibits adenylyl cyclase (EC50 values are 120 and 261 nM for CB1 and CB2 receptors respectively) and suppresses immune cell function. Learn MoreStarting at: $149.00
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CB 13
CB 13 is a potent, orally active CB1/CB2 receptor agonist with limited brain penetration (EC50 values are 6.1 and 27.9 nM for CB1 and CB2 receptors respectively), which displays antihyperalgesic activity in a rat model of neuropathic pain with no CNS side effects. Learn MoreStarting at: $95.00
