Adrenergic Receptors
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Pronethalol hydrochloride
Pronethalol hydrochloride is a ??-adrenergic antagonist, clinically effective in the treatment of angina pectoris and some arrhythmias. Learn MoreStarting at: $69.00
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Bucindolol
Bucindolol is a non-selective β-adrenoceptor antagonist with additional α1-adrenoceptor blocking activity. Ki values are 1.61, 1.20 and 68.9 nM for β1-, β2- and α1-adrenoceptors respectively. Learn MoreStarting at: $139.00
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Oxprenolol hydrochloride
Oxprenolol hydrochloride is a non-selective β-adrenergic antagonist. Learn MoreStarting at: $59.00
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ICI 89406
ICI 89406 is a β-adrenergic antagonist and low efficacy partial agonist. Learn MoreStarting at: $91.00
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(R)-(+)-Propranolol hydrochloride
(R)-(+)-Propranolol hydrochloride is a less active enantiomer of the β-adrenoceptor antagonist propranolol. Learn MoreStarting at: $69.00
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SDZ 21009
SDZ 21009 is a β-adrenoceptor and 5-HT1A/1B receptor antagonist. pKB/pA2 values are 8.3 and 8.0 for 5-HT1A and 5-HT1B receptors respectively. Learn MoreStarting at: $135.00
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Propranolol glycol
Propranolol glycol is a metabolite of propranolol. Learn MoreStarting at: $99.00
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Propranolol hydrochloride
Propranolol hydrochloride is a β-adrenergic antagonist. Learn MoreStarting at: $59.00
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Alprenolol hydrochloride
Alprenolol hydrochloride is a β-adrenoceptor (β2 > β1 > β3) and 5-HT1A receptor antagonist. Learn MoreStarting at: $55.00
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RS 100329 hydrochloride
RS 100329 hydrochloride is a subtype-selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors), which displays 126- and 50-fold selectivity over human α1B and α1D receptors respectively. Active in vivo. Learn MoreStarting at: $119.00
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Cirazoline hydrochloride
Cirazoline hydrochloride is a selective α1 agonist. Learn MoreStarting at: $90.00
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RS 17053 hydrochloride
Ro 60-0175 fumarate is a potent, selective 5-HT2 receptor agonist; shows selectivity for the 5-HT2C subtype (pKi values are 9, 7.5, 5.4, 5.2 and 5.6 for human 5-HT2C, 2A, 1A, 6 and 7 receptors respectively). Learn MoreStarting at: $95.00
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WB 4101 hydrochloride
WB 4101 hydrochloride is an α1A-adrenergic selective antagonist. Learn MoreStarting at: $89.00
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(R)-(-)-Phenylephrine hydrochloride
(R)-(-)-Phenylephrine hydrochloride is an α1-adrenoceptor agonist. Learn MoreStarting at: $49.00
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Terazosin hydrochloride
Terazosin hydrochloride is an α1- and α2B-adrenoceptor antagonist with Ki values of 3.3, 0.7, 1.1, 7.7, 1510 and 78.2 nM for α1A, α1B, α1D, α2B, α2A and α2C receptors respectively. Learn MoreStarting at: $70.00
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Urapidil hydrochloride
Urapidil hydrochloride is an α1-adrenoceptor antagonist and 5-HT1A receptor agonist. Learn MoreStarting at: $99.00
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Alfuzosin hydrochloride
Alfuzosin hydrochloride is a uro-selective α1 adrenoceptor antagonist that inhibits increases in intraurethral pressure caused by phenylephrine-induced contraction by 81% with minor cardiovascular effects. Learn MoreStarting at: $69.00
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AH 11110 hydrochloride
AH 11110 hydrochloride is a subtype-selective ligand for the α1B-adrenoceptor. Learn MoreStarting at: $110.00
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Rec 15/2615 dihydrochloride
Rec 15/2615 dihydrochlorideelective is a α1B-adrenoceptor antagonist (Ki values are 0.3, 1.9 and 2.6 nM at human α1B, α1A and α1D receptors respectively). Learn MoreStarting at: $110.00
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Tamsulosin hydrochloride
Tamsulosin hydrochloride is a selective α1A-adrenoceptor antagonist (pKi values are 9.97, 9.64 and 8.86 for α1A, α1B and α1D subtypes respectively). Learn MoreStarting at: $110.00