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Transporters
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WAY 213613
WAY 213613 is a potent, non-substrate inhibitor of EAAT2 (GLT-1) that displays > 44-fold selectivity over EAAT1 and EAAT3. Learn MoreStarting at: $139.00
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cis-ACBD
cis-ACBD is a potent, competitive and selective inhibitor of glutamate uptake. Learn MoreStarting at: $99.00
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L-(-)-threo-3-Hydroxyaspartic acid
L-(-)-threo-3-Hydroxyaspartic acid is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn MoreStarting at: $149.00
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L-trans-2,4-PDC
L-trans-2,4-PDC is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn MoreStarting at: $115.00
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(±)-threo-3-Methylglutamic acid
(±)-threo-3-Methylglutamic acid is a potent blocker of glutamate transport. Learn MoreStarting at: $89.00
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Lithium carbonate
Lithium carbonate is thought to act by reducing catecholamine neurotransmitter concentration, through an effect on the Na+/K+ ATPase pump. Learn MoreStarting at: $29.00
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Dihydrokainic acid
Dihydrokainic acid is a EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake. Learn MoreStarting at: $49.00
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3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride
3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride is a potent inhibitor of dopamine uptake and transport (Ki = 11.8 nM). Learn MoreStarting at: $75.00
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JHW 007 hydrochloride
JHW 007 hydrochloride is a dopamine uptake inhibitor which displays high affinity for the dopamine transporter (DAT) (Ki = 25 nM compared to 1330 and 1730 for NET and SERT respectively), and suppresses the effects of cocaine administration in a dose-dependent manner. Learn MoreStarting at: $120.00
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3-CPMT
3-CPMT binds with high affinity to the dopamine transporter (Ki = 30 nM) and blocks re-uptake of dopamine. Learn MoreStarting at: $50.00
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Mephedrone hydrochloride
Mephedrone hydrochloride Inhibits striatal dopamine uptake and hippocampal 5-HT uptake in synaptosomes (IC50 values are 467 and 558 nM respectively). Learn MoreStarting at: $95.00
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BTCP maleate
BTCP maleate is a potent dopamine re-uptake inhibitor with a behavioral profile different from that of PCP and similar to that of cocaine. Learn MoreStarting at: $95.00
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Zoniporide dihydrochloride
Zoniporide dihydrochloride is a sodium-hydrogen exchanger isoform 1 (NHE1) inhibitor that displays selectivity over other NHE isoforms (Ki values are 14, 2200 and 220000 nM for human NHE1, human NHE2 and rat NHE3 respectively). Learn MoreStarting at: $140.00
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Threo-methylphenidate hydrochloride
Psychomotor stimulant. Inhibitor of dopamine and noradrenalin transporters that increases the extracellular concentration of dopamine and noradrenalin. Learn MoreStarting at: $85.00
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GBR 13069 dihydrochloride
GBR 13069 dihydrochloride is a potent inhibitor of dopamine uptake with an IC50 value of 40 nM. Learn MoreStarting at: $89.00
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GBR 12783 dihydrochloride
GBR 12783 dihydrochloride is a potent and selective inhibitor of dopamine uptake with IC50 value of 1.8 nM for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes. Learn MoreStarting at: $99.00
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Cocaine hydrochloride
Cocaine hydrochloride, a competitive inhibitor of monoamine neurotransmitter transporters, inhibits dopamine (DAT), serotonin (SERT) and noradrenalin (NET) transporters with Ki values are 267, 392 and 872 nM respectively. Learn MoreStarting at: $79.00
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Nomifensine
Nomifensine is a potent inhibitor of noradrenalin and dopamine uptake (Ki values are 4.7, 26 and 4000 nM for inhibition of noradrenalin, dopamine and 5-HT uptake respectively, in rat brain), which increases central dopamine levels in rats following systemic administration. Learn MoreStarting at: $79.00
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Bupropion hydrochloride
Bupropion hydrochloride is a non-selective inhibitor of dopamine and noradrenalin transporters (Ki values are 1.4, 2.8 and 45 μM for NET, DAT and SERT transporters respectively), which also inhibits neuronal nicotinic acetylcholine receptors. Learn MoreStarting at: $99.00
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(-)-5'-DMH-CBD
(-)-5'-DMH-CBD is an anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable, which displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Learn MoreStarting at: $149.00
