Free Fatty Acid Receptors
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TUG 424
TUG 424 is an agonist of the free fatty acid receptor FFA1 (GPR40) (EC50 = 32 nM), which enhances glucose-stimulated insulin secretion in INS-1E cells at 100 nM. Learn MoreStarting at: $110.00
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4-CMTB
4-CMTB is a free fatty acid receptor FFA2 agonist (pEC50 = 6.38) and positive allosteric modulator, which binds at a site distinct from the orthosteric site; modulates the activity of short-chain fatty acids at FFA2 via the FFA2 second extracellular loop (ECL2). Learn MoreStarting at: $105.00
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MEDICA 16
MEDICA 16 is a free fatty acid 1 (FFA1/GPR40) receptor agonist that reduces intracellular triacylglycerol levels in muscle and inhibits lipogenesis and increases insulin sensitivity in rodents in vivo. Learn MoreStarting at: $115.00