Estrogen (GPR30) Receptors
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G-15
G-15 is a high affinity and selective GPR30 receptor antagonist (Ki = 20 nM) that displays no affinity for ERα and ERβ at concentrations up to 10 μM. Learn MoreStarting at: $120.00
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G-36
G-36 is an antagonist of GPR30 which selectively inhibits estrogen-mediated activation of PI3-K by GPR30. Learn MoreStarting at: $135.00
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G-1
G-1 is a potent and selective GPR30 receptor agonist that increases cytosolic Ca2+ and inhibits migration of SKBr3 cells and MCF-7 cells in response to chemoattractants with IC50 values of 0.7 and 1.6 nM respectively in vitro. Learn MoreStarting at: $139.00