You have no items in your shopping cart.
Dopamine Receptors
-
NGB 2904
NGB 2904 is a potent and selective dopamine D3 receptor antagonist (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4, D1 and D5 receptors respectively). Learn MoreStarting at: $135.00
-
PNU 177864 hydrochloride
PNU 177864 hydrochloride is a highly selective dopamine D3 receptor antagonist which induces phospholipidosis and exhibits antischizophrenic activity in vivo. Learn MoreStarting at: $109.00
-
7-Hydroxy-PIPAT maleate
8-Hydroxy-PIPAT oxalate is a high affinity 5-HT1A receptor agonist (Kd = 0.38 nM). Learn MoreStarting at: $120.00
-
PG 01037 dihydrochloride
PG 01037 dihydrochloride is a Dopamine D3 receptor antagonist with 133-fold selectivity for D3 over D2 receptors in vitro (Ki values are 0.70, 93.3 and 375 nM for D3, D2 and D4 receptors respectively). Learn MoreStarting at: $139.00
-
7-Hydroxy-DPAT hydrobromide
7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist. Learn MoreStarting at: $59.00
-
U 99194 maleate
U 99194 maleateis a potent, selective D3 antagonist. Learn MoreStarting at: $109.00
-
Sumanirole maleate
Sumanirole maleate is a high affinity D2 receptor agonist (EC50 values are between 17 and 75 nM in cell-based assays) and displays >200-fold selectivity for the D2 receptor against other dopamine receptor subtypes (Ki values are 9.0, 1940, >2190 and >7140 for D2, D3, D4 and D1 receptors respectively). Learn MoreStarting at: $130.00
-
(+)-UH 232 maleate
(+)-UH 232 maleate is a D2 antagonist (Ki = 72.7 nM in a ligand binding assay; apparent KB = 14.5 nM in a cAMP accumulation assay), which displays preferential activity at central dopamine autoreceptors. Learn MoreStarting at: $109.00
-
Prochlorperazine dimaleate
Prochlorperazine dimaleate is a D2 receptor antagonist. Learn MoreStarting at: $55.00
-
LY 379268 disodium salt
LY 379268 disodium salt is a sodium salt of LY 379268, a highly selective group II mGlu receptor agonist. Learn MoreStarting at: $295.00
-
SKF 77434 hydrobromide
SKF 77434 hydrobromide is a selective dopamine D1-like receptor partial agonist (IC50 values are 19.7 and 2425 nM for binding to D1-like and D2-like receptors respectively). Learn MoreStarting at: $79.00
-
Dihydrexidine hydrochloride
Dihydrexidine hydrochloride is a potent, full efficacy dopamine D1 agonist which shows no agonist activity at peripheral D2 receptors or adrenoceptors at doses which cause maximal stimulation of D1 sites. Learn MoreStarting at: $95.00
-
SCH 23390 hydrochloride
SCH 23390 hydrochloride is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types respectively). Learn MoreStarting at: $90.00
-
A 68930 hydrochloride
A 68930 hydrochloride is a potent and selective D1-like dopamine receptor agonist (EC50 values are 2.1 and 3910 nM for D1-like and D2-like receptors respectively). Learn MoreStarting at: $115.00
-
A 77636 hydrochloride
A 77636 hydrochloride is a potent and selective dopamine D1-like receptor agonist (pEC50 values are 8.97 and < 5 for D1-like and D2-like receptors respectively), which displays anti-Parkinsonian activity following oral administration in vivo. Learn MoreStarting at: $140.00
-
LE 300
LE 300 is a potent and selective dopamine D1 receptor antagonist (Ki values are 0.08 - 1.9 nM and 6 - 45 nM for D1 and D2 receptors respectively), which also displays moderate affinity for the 5-HT2A receptor (Ki = 20 nM). Active in vivo. Learn MoreStarting at: $139.00
-
CY 208-243
CY 208-243 is a centrally active dopamine D1 receptor agonist, selective over D2 receptor sites, which stimulates adenylate cyclase in rat striatal homogenates with an EC50 of 125 nM, that exerts antiParkinsonian activity in animal models. Learn MoreStarting at: $139.00
-
SKF 81297 hydrobromide
SKF 81297 hydrobromide is a dopamine D1-like receptor agonist. Learn MoreStarting at: $149.00
-
SKF 83822 hydrobromide
SKF 83822 hydrobromide is a high affinity, selective dopamine D1-like receptor agonist. Learn MoreStarting at: $139.00
-
SKF 83959 hydrobromide
SKF 83959 hydrobromide is a dopamine D1-like receptor partial agonist that act as an antagonist in vivo, producing anti-Parkinsonian effects and antagonizing the behavioral effects of cocaine. Learn MoreStarting at: $139.00
