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Search results for 'inhibitor'
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H-9 dihydrochloride
H-9 dihydrochloride is a protein kinase inhibitor that inhibits PKA, PKG, CaMK II, PKC, casein kinase I and casein kinase II. Learn MoreStarting at: $89.00
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TCS 2312
TCS 2312 is a potent and selective checkpoint kinase 1 (chk1) inhibitor that enhances the cell killing activity of Gemcitabine in breast and prostate cancer cell lines and displays antiproliferative effects in vitro. Learn MoreStarting at: $139.00
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YM 244769
YM 244769 is an inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX) that inhibits Na+-dependent 45Ca2+ uptake with IC50 values of 18, 68 and 96 nM for CCL39 cells transfected with NCX3, NCX1 and NCX2 respectively. Learn MoreStarting at: $125.00
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RHC 80267
RHC 80267 is an inhibitor of diacylglycerol lipase that potentiates acetylcholine evoked relaxation in mesenteric arteries by the inhibition of cholinesterase activity. Learn MoreStarting at: $99.00
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Nafamostat mesylate
Nafamostat mesylate is a broad spectrum serine protease inhibitor that reduces eosinophil infiltration, mast cell activation and airway responsiveness in a murine model of asthma. Learn MoreStarting at: $45.00
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CI 898 trihydrochloride
CI 898 trihydrochloride is a potent lipophilic inhibitor of dihydrofolate reductase (DHFR) that inhibits protozoal, bacterial and human DHFR with IC50 values of 1.4, 6.1 and 3.2 nM respectively. Learn MoreStarting at: $139.00
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Nefazodone hydrochloride
Nefazodone hydrochloride is a serotonin 5-HT2A receptor antagonist (Ki = 5.8 nM) and inhibitor of serotonin and noradrenalin uptake (IC50 values are 290 and 300 nM respectively). Learn MoreStarting at: $89.00
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Moexipril hydrochloride
Moexipril hydrochloride is an angiotensin-converting enzyme (ACE) inhibitor that decreases mean blood pressure in the spontaneous hypertensive rat (SHR) and also blocks degradation of bradykinin into inactive metabolites. Learn MoreStarting at: $109.00
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NSC 33994
NSC 33994 is a selective inhibitor of JAK2 with an IC50 value of 60 nM. Learn MoreStarting at: $139.00
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10Z-Hymenialdisine
10Z-Hymenialdisine is a pan kinase inhibitor that inhibits NF-κB activation and blocks IL-8 production in U937 cells with IC50 values of 1-2 and 0.34-0.48 μM respectively. Learn MoreStarting at: $259.00
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Cilastatin sodium
Cilastatin sodium is a dipeptidase inhibitor that inhibits metabolism of LTD4 to LTE4 and the hydrolysis of β-lactam antibiotics. Learn MoreStarting at: $89.00
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N-Nonyldeoxynojirimycin
N-Nonyldeoxynojirimycin is a glucosidase inhibitor that inhibits liver glycogen breakdown in vivo. Learn MoreStarting at: $139.00
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Concanamycin A
Concanamycin A is a specific inhibitor of V-type (vacuolar) H+-ATPase that blocks cell surface expression of virus envelope glycoproteins without affecting synthesis and exhibits cytotoxicity in several cell lines. Learn MoreStarting at: $99.00
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ML 130
ML 130 is a potent and selective inhibitor of NOD1 that inhibits NOD1-induced NF-κB activation in HEK293 cells with no cytotoxicity. Learn MoreStarting at: $119.00
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Castanospermine
Castanospermine is a potent inhibitor of α- and β-glucosidases that inhibits HIV syncytium formation and replication. Learn MoreStarting at: $69.00
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Sertraline hydrochloride
Sertraline hydrochloride is a potent, orally active selective serotonin re-uptake inhibitor (SSRI). Learn MoreStarting at: $109.00
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BIBU 1361 dihydrochloride
BIBU 1361 dihydrochloride is a potent inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase that inhibits growth of established human xenografts in athymic mice. Learn MoreStarting at: $85.00
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SA 47
SA 47 is a selective inhibitor of fatty acid amide hydrolase (FAAH) that exhibits greater selectivity for FAAH than URB 597 against multiple carboxylesterases. Learn MoreStarting at: $109.00
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PSB 069
PSB 069 is a non-selective nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitor. Learn MoreStarting at: $109.00
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Trequinsin hydrochloride
Trequinsin hydrochloride is an extremely potent inhibitor of cGMP-inhibited phosphodiesterase that inhibits arachidonic acid-induced aggregation of human platelets. Learn MoreStarting at: $199.00
