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Search results for 'inhibit'
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KD 5170
KD 5170 is a histone deacetylase (HDAC) inhibitor that exhibits broad spectrum inhibition of HDAC classes I and II in assays using purified recombinant human isoforms. Learn MoreStarting at: $139.00
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NSC 95397
NSC 95397 is a potent and selective irreversible inhibitor of Cdc25 dual specificity phosphatases that displays 125 - 180-fold selectivity over VH1-related dual-specificity phosphatase and protein tyrosine phosphatase 1b. Learn MoreStarting at: $139.00
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TC-H 106
TC-H 106 is a class I histone deacetylase (HDAC) inhibitor with IC50 values of 150, 370, 760 and 5000 nM for HDAC1, HDAC3, HDAC2 and HDAC8 respectively. Learn MoreStarting at: $125.00
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MDL 72527
MDL 72527 is a polyamine oxidase (POA) inhibitor that displays anticancer and neuroprotective activity in vivo. Learn MoreStarting at: $109.00
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R 59022
R 59022 is a diacylglycerol (DAG) kinase inhibitor with an IC50 value of 2.8 μM. Learn MoreStarting at: $105.00
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KC7F2
KC7F2 is an inhibitor of HIF-1α that reduces phosphorylation of eIF4E binding protein 1 (4EBP1) and p70 S6K in hypoxic conditions. Learn MoreStarting at: $69.00
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AMTB hydrochloride
AMTB hydrochloride is a TRPM8 channel blocker that inhibits icilin- induced TRPM8 channel activation in a rat model. Learn MoreStarting at: $139.00
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KU 60019
KU 60019 is a potent ATM kinase inhibitor with an IC50 value of 6.3 nM. Learn MoreStarting at: $189.00
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(±)-MDMA hydrochloride
(±)-MDMA hydrochloride is a hallucinogenic compound that inhibits 5-HT and dopamine uptake. Learn MoreStarting at: $105.00
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Zatebradine hydrochloride
Zatebradine hydrochloride is a bradycardic agent that produces use-dependent inhibition of hyperpolarization-activated current If (HCN channel) in sinoatrial node cells and Purkinje fibres. Learn MoreStarting at: $109.00
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GPi 688
GPi 688 is an allosteric glycogen phosphorylase inhibitor that inhibits glucagon-mediated hyperglycemia in vivo in the rat. Learn MoreStarting at: $179.00
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TC-I 15
TC-I 15 is a potent α2β1 integrin inhibitor. IC50 values for the inhibition of human platelet adhesion to type I collagen are 12 and 715 nM for platelets under static conditions and under flow, respectively. Learn MoreStarting at: $169.00
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Benidipine hydrochloride
Benidipine hydrochloride is an orally active antihypertensive agent that inhibits L-, N- and T-type Ca2+ channels and also inhibits aldosterone-induced mineralocorticoid receptor activation. Learn MoreStarting at: $109.00
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Noscapine hydrochloride
Noscapine hydrochloride is an opioid alkaloid that inhibits carbachol-stimulated phosphoinositol turnover and enhances forskolin-stimulated cAMP increases in CNS tissues. Learn MoreStarting at: $75.00
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A 83-01
A 83-01 is a selective inhibitor of TGF-β type I receptor ALK5 kinase, type I activin/nodal receptor ALK4 and type I nodal receptor ALK7 . Learn MoreStarting at: $135.00
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CGK 733
CGK 733 is originally defined as a selective inhibitor of ATR and ATM kinases that decreases p21CIP1 levels in premature senescent MCF-7 and HCT-116 cells. Learn MoreStarting at: $105.00
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NU 1025
NU 1025 is a novel, potent inhibitor of poly(ADP-ribose) polymerase (PARP). Learn MoreStarting at: $105.00
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FPA 124
FPA 124 is an Akt/PKB inhibitor that inhibits cell proliferation in various cancer cell lines in vitro and decreases NF-κB activity and tumor load in vivo. Learn MoreStarting at: $125.00
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AT 101
AT101, a natural product from cottonseed with a BH3-mimetic structure, was identified as a small molecule inhibitor of Bcl-2/Bcl-xL/Mcl-1 that potently induces apoptosis in various cancer cell lines. Learn MoreStarting at: $105.00
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(±)-Clopidogrel hydrochloride
(±)-Clopidogrel hydrochloride is a selective, high affinity P2Y12 receptor antagonist that inhibits ADP-induced platelet aggregation. Learn MoreStarting at: $99.00
