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Search results for 'inhibitor'
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(-)-5'-DMH-CBD
(-)-5'-DMH-CBD is an anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable, which displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Learn MoreStarting at: $149.00
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(±)-McN 5652
(±)-McN 5652 is a potent, high affinity serotonin re-uptake inhibitor; selective in viv, and displays moderate selectivity over noradrenalin and dopamine re-uptake in vitro (Ki values are 0.68, 2.9 and 36.8 nM for inhibition of serotonin, noradrenalin and dopamine uptake respectively in rat brain synaptosomes). Learn MoreStarting at: $139.00
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SD 1008
SD 1008 is a JAK2/STAT3 signaling pathway inhibitor, which inhibits activation of STAT3, JAK2 and Src. Learn MoreStarting at: $109.00
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PF 750
PF 750 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor that displays no activity at a range of other serine hydrolases. Learn MoreStarting at: $149.00
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SID 26681509
SID 26681509 is a potent and reversible human cathepsin L inhibitor with an IC50 value of 56 nM. Learn MoreStarting at: $149.00
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PF 04217903 mesylate
PF 04217903 mesylate is a highly selective, high affinity c-Met inhibitor that displays >1000-fold selectivity for c-Met over a panel of 208 kinases. Learn MoreStarting at: $189.00
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TCS HDAC6 20b
TCS HDAC6 20b is a selective inhibitor of histone deacetylase 6 (HDAC6) that inhibits HCT116 growth in combination with taxol. Learn MoreStarting at: $149.00
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WWL 70
WWL 70 is a potent inhibitor of α/β-hydrolase domain 6 (ABHD6) with an IC50 of 70 nM. Learn MoreStarting at: $75.00
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JNJ 28871063 hydrochloride
JNJ 28871063 hydrochloride is a potent and selective ErbB receptor family inhibitor with IC50 values of 21, 22 and 38 nM for ErbB4, EGFR and ErbB2 respectively. Learn MoreStarting at: $139.00
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PHA 767491 hydrochloride
PHA 767491 hydrochloride is a potent, ATP-competitive dual cdc7/cdk9 inhibitor with IC50 valuesof 10 and 34 nM respectively. Learn MoreStarting at: $99.00
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PI 828
PI 828 is a PI 3-Kinase inhibitor with IC50 values of 0.098, 0.183, 0.227 and 1.967 μM for p110β, p110α, p110δ and p110γ respectively. Learn MoreStarting at: $69.00
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KD 5170
KD 5170 is a histone deacetylase (HDAC) inhibitor that exhibits broad spectrum inhibition of HDAC classes I and II in assays using purified recombinant human isoforms. Learn MoreStarting at: $139.00
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NSC 95397
NSC 95397 is a potent and selective irreversible inhibitor of Cdc25 dual specificity phosphatases that displays 125 - 180-fold selectivity over VH1-related dual-specificity phosphatase and protein tyrosine phosphatase 1b. Learn MoreStarting at: $139.00
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TC-H 106
TC-H 106 is a class I histone deacetylase (HDAC) inhibitor with IC50 values of 150, 370, 760 and 5000 nM for HDAC1, HDAC3, HDAC2 and HDAC8 respectively. Learn MoreStarting at: $125.00
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MDL 72527
MDL 72527 is a polyamine oxidase (POA) inhibitor that displays anticancer and neuroprotective activity in vivo. Learn MoreStarting at: $109.00
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R 59022
R 59022 is a diacylglycerol (DAG) kinase inhibitor with an IC50 value of 2.8 μM. Learn MoreStarting at: $105.00
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KC7F2
KC7F2 is an inhibitor of HIF-1α that reduces phosphorylation of eIF4E binding protein 1 (4EBP1) and p70 S6K in hypoxic conditions. Learn MoreStarting at: $69.00
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KU 60019
KU 60019 is a potent ATM kinase inhibitor with an IC50 value of 6.3 nM. Learn MoreStarting at: $189.00
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GPi 688
GPi 688 is an allosteric glycogen phosphorylase inhibitor that inhibits glucagon-mediated hyperglycemia in vivo in the rat. Learn MoreStarting at: $179.00
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TC-I 15
TC-I 15 is a potent α2β1 integrin inhibitor. IC50 values for the inhibition of human platelet adhesion to type I collagen are 12 and 715 nM for platelets under static conditions and under flow, respectively. Learn MoreStarting at: $169.00
